XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa MAP3K5
DIkGDNVLINTYSGVLK
Lys2
1.8
10
uM
XMD-12 PC-3 M3K2,MAP3K3
DIkGANILR
Lys2
18.0
10
uM
XMD-12 HeLa M3K2,MAP3K3
DIkGANILR
Lys2
39.6
10
uM
XMD-12 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
-0.6
10
uM
XMD-12 HeLa MAP3K4
DIkGANIFLTSSGLIK
Lys2
-23.3
10
uM
XMD-12 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
52.3
10
uM
XMD-12 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
28.9
10
uM
XMD-12 PC-3 MST1,MST2
DIkAGNILLNTEGHAK
Lys2
39.1
10
uM
XMD-12 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
28.6
10
uM
XMD-12 HeLa MST3
DIkAANVLLSEHGEVK
Lys2
15.0
10
uM
XMD-12 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
-13.9
10
uM
XMD-12 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
85.4
10
uM
XMD-12 PC-3 AGK
ATVFLNPAACkGK
ATP
-6.7
10
uM
XMD-12 PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
1.9
10
uM
XMD-12 HeLa LATS1
ALYATkTLR
Lys1
-36.0
10
uM
XMD-12 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
0.5
10
uM