XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 PC-3 CDK16
LTDNLVALkEIR
Lys1
-11.1
10
uM
XMD-12 PC-3 CDK14
LVALkVIR
Lys1
1.1
10
uM
XMD-12 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
1.1
10
uM
XMD-12 HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
10.9
10
uM
XMD-12 HeLa MAP2K6
DVkPSNVLINALGQVK
Lys2
-10.4
10
uM
XMD-12 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-10.2
10
uM
XMD-12 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-10.1
10
uM
XMD-12 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-10.0
10
uM
XMD-12 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
-0.6
10
uM
XMD-12 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
0.5
10
uM
XMD-12 PC-3 EGFR
IPVAIkELR
Lys1
-0.3
10
uM
XMD-12 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
0.2
10
uM
XMD-12 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
0.2
10
uM
XMD-12 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD-12 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
10
uM
XMD-12 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
10
uM