XMD-12 KiNativ -- single dose experiment - Dataset (ID:20103)

 Full screen view
Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD-12 HeLa KPCI
IYAMkVVK
Lys1
-50.8
 10
uM
XMD-12 HeLa GCN2
LDGCCYAVkR
Lys1
-5.1
 10
uM
XMD-12 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
-7.6
 10
uM
XMD-12 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
12.8
 10
uM
XMD-12 HeLa PKD2
DVAVkVIDK
Lys1
5.0
 10
uM
XMD-12 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
1.9
 10
uM
XMD-12 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
27.4
 10
uM
XMD-12 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
-11.2
 10
uM
XMD-12 HeLa SYK
ISDFGLSkALR
Activation Loop
2.1
 10
uM
XMD-12 HeLa TLK1
YAAVkIHQLNK
Lys1
-23.8
 10
uM
XMD-12 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-9.3
 10
uM
XMD-12 HeLa AurB
SHFIVALkVLFK
Lys1
95.0
 10
uM
XMD-12 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
23.7
 10
uM
XMD-12 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-1.3
 10
uM
XMD-12 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
11.2
 10
uM
XMD-12 HeLa ILK
WQGIVVkVLK
Lys1
-4.0
 10
uM