XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD8-85 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -26.4 | 10 | uM |
| XMD8-85 | PC-3 | IKKE,TBK1 | DIkPGNIMR | Lys2 | 1.5 | 10 | uM |
| XMD8-85 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -11.2 | 10 | uM |
| XMD8-85 | PC-3 | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | 6.5 | 10 | uM |
| XMD8-85 | PC-3 | GSK3B | DIkPQNLLLDPDTAVLK | Lys2 | 5.4 | 10 | uM |
| XMD8-85 | HeLa | GSK3A | DIkPQNLLVDPDTAVLK | Lys2 | -12.2 | 10 | uM |
| XMD8-85 | PC-3 | MAP2K4 | DIkPSNILLDR | Lys2 | -18.8 | 10 | uM |
| XMD8-85 | PC-3 | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -12.8 | 10 | uM |
| XMD8-85 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -1.8 | 10 | uM |
| XMD8-85 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -23.1 | 10 | uM |
| XMD8-85 | HeLa | NEK9 | DIkTLNIFLTK | Lys2 | -9.4 | 10 | uM |
| XMD8-85 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 14.5 | 10 | uM |
| XMD8-85 | HeLa | HPK1 | DKVSGDLVALkMVK | Lys1 | -10.1 | 10 | uM |
| XMD8-85 | PC-3 | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 9.6 | 10 | uM |
| XMD8-85 | HeLa | MARK2,MARK3 | DLkAENLLLDADMNIK | Lys2 | 4.9 | 10 | uM |
| XMD8-85 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | -5.2 | 10 | uM |
| XMD8-85 | HeLa | SLK | DLkAGNILFTLDGDIK | Lys2 | -13.0 | 10 | uM |
| XMD8-85 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 1.2 | 10 | uM |
| XMD8-85 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | -10.4 | 10 | uM |
| XMD8-85 | HeLa | Wnk1,Wnk2,Wnk3 | DLkCDNIFITGPTGSVK | Lys2 | -17.8 | 10 | uM |
| XMD8-85 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | -6.3 | 10 | uM |
| XMD8-85 | PC-3 | PKCa,PKCb | DLkLDNVMLDSEGHIK | Lys2 | -27.9 | 10 | uM |
| XMD8-85 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | 2.6 | 10 | uM |
| XMD8-85 | HeLa | BARK1 | DLkPANILLDEHGHVR | Lys2 | -22.1 | 10 | uM |
| XMD8-85 | PC-3 | CDK11,CDK8 | DLkPANILVMGEGPER | Lys2 | 6.2 | 10 | uM |