XMD8-85 KiNativ -- single dose experiment - Dataset - HMS LINCS Database

XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

<<<<

Select the entities to show:

Small molecules	Cells	Proteins

Small Molecule	Cell Line	Protein	Sequence	Labeling Site	% Inhibition	Assay compound conc	Conc unit
XMD8-85	HeLa	CDK2	DLkPQNLLINTEGAIK	Lys2	-15.8	10	uM
XMD8-85	PC-3	CDK2	DLkPQNLLINTEGAIK	Lys2	3.3	10	uM
XMD8-85	PC-3	CDK5	DLkPQNLLINR	Lys2	-21.8	10	uM
XMD8-85	PC-3	CDK5	NRETHEIVALkR	Lys1	-9.5	10	uM
XMD8-85	PC-3	CDK5	ETHEIVALkR	Lys1	-24.1	10	uM
XMD8-85	HeLa	CDK7	DLkPNNLLLDENGVLK	Lys2	-2.7	10	uM
XMD8-85	PC-3	CDK9	DMkAANVLITR	Lys2	2.1	10	uM
XMD8-85	HeLa	CHK1	DIkPENLLLDER	Lys2	-7.7	10	uM
XMD8-85	PC-3	CHK2	VAIkIISK	Lys1	14.0	10	uM
XMD8-85	PC-3	CHK2	DLkPENVLLSSQEEDCLIK	Lys2	30.3	10	uM
XMD8-85	HeLa	CHK2	DLkPENVLLSSQEEDCLIK	Lys2	16.4	10	uM
XMD8-85	PC-3	CK1d,CK1e	DVkPDNFLMGLGKK	Lys2	-12.2	10	uM
XMD8-85	PC-3	CLK2	LTHTDLkPENILFVNSDYELTYNLEK	Lys2	6.2	10	uM
XMD8-85	HeLa	CSK	VSDFGLTkEASSTQDTGKLPVK	Activation Loop	3.0	10	uM
XMD8-85	PC-3	CSK	VSDFGLTkEASSTQDTGKLPVK	Activation Loop	-13.6	10	uM
XMD8-85	HeLa	DGKA	IDPVPNTHPLLVFVNPkSGGK	ATP	-1.9	10	uM
XMD8-85	HeLa	DMPK	DIkPDNILLDR	Lys2	-13.2	10	uM
XMD8-85	PC-3	DNAPK	GHDEREHPFLVkGGEDLRQDQR	ATP	31.0	10	uM
XMD8-85	HeLa	DNAPK	GHDEREHPFLVkGGEDLRQDQR	ATP	12.3	10	uM
XMD8-85	PC-3	DNAPK	kGGSWIQEINVAEK	ATP	3.6	10	uM
XMD8-85	PC-3	eEF2K	YIkYNSNSGFVR	Protein Kinase Domain	3.8	10	uM
XMD8-85	HeLa	eEF2K	YIkYNSNSGFVR	Protein Kinase Domain	-22.1	10	uM
XMD8-85	PC-3	EGFR	ITDFGLAkLLGAEEK	Activation Loop	-1.5	10	uM
XMD8-85	PC-3	EGFR	LLGAEEKEYHAEGGkVPIK	Activation Loop	21.9	10	uM
XMD8-85	PC-3	EGFR	IPVAIkELR	Lys1	-6.8	10	uM