XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-47.0
10
uM
XMD8-85 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-3.5
10
uM
XMD8-85 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
13.1
10
uM
XMD8-85 HeLa TLK1
YAAVkIHQLNK
Lys1
-38.6
10
uM
XMD8-85 PC-3 TLK1
YAAVkIHQLNK
Lys1
-5.2
10
uM
XMD8-85 PC-3 TLK2
YVAVkIHQLNK
Lys1
5.0
10
uM
XMD8-85 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-4.3
10
uM
XMD8-85 HeLa ULK3
EVVAIkCVAK
Lys1
-13.9
10
uM
XMD8-85 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
-14.6
10
uM
XMD8-85 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
-17.8
10
uM
XMD8-85 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-7.8
10
uM
XMD8-85 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-6.3
10
uM
XMD8-85 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-17.3
10
uM
XMD8-85 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
-12.4
10
uM