XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
90.3
10
uM
XMD8-85 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
9.2
10
uM
XMD8-85 HeLa MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
-9.3
10
uM
XMD8-85 PC-3 NEK9
LGDYGLAkK
Activation Loop
-9.3
10
uM
XMD8-85 HeLa MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
-9.3
10
uM
XMD8-85 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
9.3
10
uM
XMD8-85 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-9.4
10
uM
XMD8-85 HeLa NEK9
DIkTLNIFLTK
Lys2
-9.4
10
uM
XMD8-85 PC-3 MST4,YSK1
DIkAANVLLSEQGDVK
Lys2
-9.5
10
uM
XMD8-85 PC-3 CDK5
NRETHEIVALkR
Lys1
-9.5
10
uM
XMD8-85 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
9.6
10
uM
XMD8-85 PC-3 TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
9.6
10
uM
XMD8-85 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.3
10
uM
XMD8-85 HeLa FES
LRADNTLVAVkSCR
Lys1
-9.8
10
uM