XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
3.6
10
uM
XMD8-85 PC-3 PI42C
ELPTLkDMDFLNK
ATP
20.5
10
uM
XMD8-85 PC-3 AGK
ATVFLNPAACkGK
ATP
4.6
10
uM
XMD8-85 HeLa PIK3CG
KkPLWLEFK
ATP
-13.4
10
uM
XMD8-85 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
31.0
10
uM
XMD8-85 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
-1.9
10
uM
XMD8-85 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
7.0
10
uM
XMD8-85 PC-3 ATR
FYIMMCkPK
ATP
5.4
10
uM
XMD8-85 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
1.1
10
uM
XMD8-85 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
74.4
10
uM
XMD8-85 HeLa ATR
FYIMMCkPK
ATP
-18.0
10
uM
XMD8-85 PC-3 PIK3CB
VFGEDSVGVIFkNGDDLRQDMLTLQMLR
ATP
-8.7
10
uM
XMD8-85 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
16.2
10
uM
XMD8-85 HeLa PI4KB
VPHTQAVVLNSkDK
ATP
-17.4
10
uM
XMD8-85 HeLa PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
-2.8
10
uM
XMD8-85 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
17.1
10
uM
XMD8-85 PC-3 PI4KB
VPHTQAVVLNSkDK
ATP
-1.3
10
uM
XMD8-85 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-8.2
10
uM
XMD8-85 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
3.7
10
uM
XMD8-85 HeLa MSK1,MSK2_domain1
VLGTGAYGkVFLVR
ATP Loop
-18.1
10
uM
XMD8-85 HeLa MAPKAPK3
KYAVTDDYQLSkQVLGLGVNGK
ATP Loop
-15.8
10
uM
XMD8-85 HeLa PRPK
FLSGLELVkQGAEAR
ATP Loop
-2.9
10
uM
XMD8-85 PC-3 PRPK
FLSGLELVkQGAEAR
ATP Loop
17.9
10
uM
XMD8-85 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
7.6
10
uM
XMD8-85 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
50.6
10
uM