XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 HeLa MK14
QELNkTIWEVPER
Other
-19.8
10
uM
XMD8-85 PC-3 MK11
QELNkTVWEVPQR
Other
6.3
10
uM
XMD8-85 PC-3 ROCK1
kLQLELNQER
Other
-11.7
10
uM
XMD8-85 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
8.2
10
uM
XMD8-85 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
16.7
10
uM
XMD8-85 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
70.1
10
uM
XMD8-85 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-22.1
10
uM
XMD8-85 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
27.9
10
uM
XMD8-85 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
9.2
10
uM
XMD8-85 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
28.6
10
uM
XMD8-85 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-0.8
10
uM
XMD8-85 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-131.3
10
uM
XMD8-85 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
3.8
10
uM
XMD8-85 HeLa PAN3
VMDPTkILITGK
-7.7
10
uM