XMD8-85 KiNativ -- single dose experiment - Dataset (ID:20101)

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  • 1 to 25 of 239 records
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD8-85 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
9.0
10
uM
XMD8-85 HeLa SYK
ISDFGLSkALR
Activation Loop
-12.8
10
uM
XMD8-85 PC-3 MET
DMYDkEYYSVHNK
Activation Loop
15.3
10
uM
XMD8-85 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-1.5
10
uM
XMD8-85 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
10.6
10
uM
XMD8-85 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-12.5
10
uM
XMD8-85 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-13.6
10
uM
XMD8-85 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-2.0
10
uM
XMD8-85 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
21.9
10
uM
XMD8-85 PC-3 NEK9
LGDYGLAkK
Activation Loop
-9.3
10
uM
XMD8-85 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
-22.8
10
uM
XMD8-85 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
13.5
10
uM
XMD8-85 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
-25.7
10
uM
XMD8-85 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
17.7
10
uM
XMD8-85 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
-63.6
10
uM
XMD8-85 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
3.0
10
uM
XMD8-85 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
-21.5
10
uM
XMD8-85 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-7.8
10
uM
XMD8-85 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
4.2
10
uM
XMD8-85 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
6.2
10
uM
XMD8-85 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
-18.1
10
uM
XMD8-85 HeLa NEK9
LGDYGLAkK
Activation Loop
-6.5
10
uM
XMD8-85 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
-27.9
10
uM
XMD8-85 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
-47.0
10
uM
XMD8-85 HeLa PIK3C3
TEDGGKYPVIFkHGDDLR
ATP
74.4
10
uM
  • Page 1 of 10
  • 1 to 25 of 239 records