JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
14.8
 10
uM
JWE-035 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
6.7
 10
uM
JWE-035 PC-3 CDK5
DLkPQNLLINR
Lys2
13.4
 10
uM
JWE-035 PC-3 CDK5
NRETHEIVALkR
Lys1
34.0
 10
uM
JWE-035 PC-3 CDK5
ETHEIVALkR
Lys1
54.2
 10
uM
JWE-035 HeLa CDK7
DLkPNNLLLDENGVLK
Lys2
54.2
 10
uM
JWE-035 PC-3 CDK9
DMkAANVLITR
Lys2
4.2
 10
uM
JWE-035 HeLa CHK1
DIkPENLLLDER
Lys2
-6.0
 10
uM
JWE-035 PC-3 CHK2
VAIkIISK
Lys1
42.7
 10
uM
JWE-035 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
-1.7
 10
uM
JWE-035 HeLa CHK2
DLkPENVLLSSQEEDCLIK
Lys2
5.9
 10
uM
JWE-035 PC-3 CK1d,CK1e
DVkPDNFLMGLGKK
Lys2
-1.7
 10
uM
JWE-035 PC-3 CK2a2
DVkPHNVMIDHQQK
Lys2
31.6
 10
uM
JWE-035 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
20.4
 10
uM
JWE-035 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
3.2
 10
uM
JWE-035 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-6.1
 10
uM
JWE-035 HeLa DGKA
IDPVPNTHPLLVFVNPkSGGK
ATP
-0.7
 10
uM
JWE-035 HeLa DMPK
DIkPDNILLDR
Lys2
-5.1
 10
uM
JWE-035 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
4.9
 10
uM
JWE-035 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
29.7
 10
uM
JWE-035 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
66.4
 10
uM
JWE-035 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.3
 10
uM
JWE-035 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.9
 10
uM
JWE-035 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
5.8
 10
uM
JWE-035 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-6.9
 10
uM