JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
66.4
 10
uM
JWE-035 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
6.7
 10
uM
JWE-035 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
6.8
 10
uM
JWE-035 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
68.1
 10
uM
JWE-035 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-6.9
 10
uM
JWE-035 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.1
 10
uM
JWE-035 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
71.7
 10
uM
JWE-035 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
7.2
 10
uM
JWE-035 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
 10
uM
JWE-035 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
7.3
 10
uM
JWE-035 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
75.6
 10
uM
JWE-035 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
75.7
 10
uM
JWE-035 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
76.9
 10
uM
JWE-035 PC-3 RON
IQCAIkSLSR
Lys1
7.7
 10
uM
JWE-035 PC-3 EGFR
IPVAIkELR
Lys1
7.8
 10
uM
JWE-035 PC-3 PI42C
ELPTLkDMDFLNK
ATP
78.9
 10
uM
JWE-035 HeLa MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
7.9
 10
uM
JWE-035 HeLa MK14
QELNkTIWEVPER
Other
7.9
 10
uM
JWE-035 PC-3 MAP2K3
DVkPSNVLINK
Lys2
7.9
 10
uM
JWE-035 HeLa AurB
SHFIVALkVLFK
Lys1
80.4
 10
uM
JWE-035 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
-8.1
 10
uM
JWE-035 HeLa ATR
FYIMMCkPK
ATP
8.1
 10
uM
JWE-035 HeLa ULK3
EVVAIkCVAK
Lys1
8.2
 10
uM
JWE-035 HeLa PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
83.0
 10
uM
JWE-035 PC-3 EPHA2
EVPVAIkTLK
Lys1
8.4
 10
uM