JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 ROCK1,ROCK2
DVkPDNMLLDK
Lys2
-1.5
10
uM
JWE-035 PC-3 MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
15.9
10
uM
JWE-035 PC-3 NEK9
DIkTLNIFLTK
Lys2
15.9
10
uM
JWE-035 HeLa MAP2K3
DVkPSNVLINK
Lys2
-1.6
10
uM
JWE-035 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
16.0
10
uM
JWE-035 PC-3 LOK
DLkAGNVLMTLEGDIR
Lys2
16.0
10
uM
JWE-035 PC-3 EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
16.2
10
uM
JWE-035 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
16.8
10
uM
JWE-035 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
16.9
10
uM
JWE-035 PC-3 CK1d,CK1e
DVkPDNFLMGLGKK
Lys2
-1.7
10
uM
JWE-035 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
-1.7
10
uM
JWE-035 PC-3 CHK2
DLkPENVLLSSQEEDCLIK
Lys2
-1.7
10
uM
JWE-035 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
17.1
10
uM
JWE-035 HeLa MST3
DIkAANVLLSEHGEVK
Lys2
17.5
10
uM
JWE-035 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
18.0
10
uM
JWE-035 PC-3 GCN2
LDGCCYAVkR
Lys1
18.1
10
uM
JWE-035 PC-3 AGK
ATVFLNPAACkGK
ATP
-18.2
10
uM
JWE-035 PC-3 ROCK1
kLQLELNQER
Other
18.7
10
uM
JWE-035 HeLa NEK9
LGDYGLAkK
Activation Loop
-19.5
10
uM
JWE-035 HeLa NEK1
DIkSQNIFLTK
Lys2
-19.6
10
uM
JWE-035 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
19.9
10
uM
JWE-035 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
19.9
10
uM
JWE-035 HeLa TAO1,TAOK3
DIkAGNILLTEPGQVK
Lys2
-2.0
10
uM
JWE-035 PC-3 SRC
VAIkTLKPGTMSPEAFLQEAQVMK
Lys1
-2.0
10
uM
JWE-035 HeLa BTK
GQYDVAIkMIK
Lys1
2.0
10
uM