JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JWE-035 | PC-3 | ROCK1,ROCK2 | DVkPDNMLLDK | Lys2 | -1.5 | 10 | uM |
JWE-035 | PC-3 | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 15.9 | 10 | uM |
JWE-035 | PC-3 | NEK9 | DIkTLNIFLTK | Lys2 | 15.9 | 10 | uM |
JWE-035 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | -1.6 | 10 | uM |
JWE-035 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 16.0 | 10 | uM |
JWE-035 | PC-3 | LOK | DLkAGNVLMTLEGDIR | Lys2 | 16.0 | 10 | uM |
JWE-035 | PC-3 | EPHB4 | FLEENSSDPTYTSSLGGkIPIR | Activation Loop | 16.2 | 10 | uM |
JWE-035 | PC-3 | EphA1 | LLDDFDGTYETQGGkIPIR | Activation Loop | 16.8 | 10 | uM |
JWE-035 | HeLa | RSK2_domain2 | SkRDPTEEIEILLR | Protein Kinase Domain | 16.9 | 10 | uM |
JWE-035 | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | -1.7 | 10 | uM |
JWE-035 | HeLa | IKKA | DLkPENIVLQDVGGK | Lys2 | -1.7 | 10 | uM |
JWE-035 | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -1.7 | 10 | uM |
JWE-035 | PC-3 | MST1 | ETGQIVAIkQVPVESDLQEIIK | Lys1 | 17.1 | 10 | uM |
JWE-035 | HeLa | MST3 | DIkAANVLLSEHGEVK | Lys2 | 17.5 | 10 | uM |
JWE-035 | PC-3 | M4K3 | NVNTGELAAIkVIK | Lys1 | 18.0 | 10 | uM |
JWE-035 | PC-3 | GCN2 | LDGCCYAVkR | Lys1 | 18.1 | 10 | uM |
JWE-035 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -18.2 | 10 | uM |
JWE-035 | PC-3 | ROCK1 | kLQLELNQER | Other | 18.7 | 10 | uM |
JWE-035 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | -19.5 | 10 | uM |
JWE-035 | HeLa | NEK1 | DIkSQNIFLTK | Lys2 | -19.6 | 10 | uM |
JWE-035 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.9 | 10 | uM |
JWE-035 | PC-3 | IRAK1 | AIQFLHQDSPSLIHGDIkSSNVLLDER | Lys2 | 19.9 | 10 | uM |
JWE-035 | HeLa | TAO1,TAOK3 | DIkAGNILLTEPGQVK | Lys2 | -2.0 | 10 | uM |
JWE-035 | PC-3 | SRC | VAIkTLKPGTMSPEAFLQEAQVMK | Lys1 | -2.0 | 10 | uM |
JWE-035 | HeLa | BTK | GQYDVAIkMIK | Lys1 | 2.0 | 10 | uM |