JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 HeLa PLK1
DLkLGNLFLNEDLEVK
Lys2
-1.2
10
uM
JWE-035 PC-3 PDK1
EYAIkILEK
Lys1
12.1
10
uM
JWE-035 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
12.1
10
uM
JWE-035 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
12.2
10
uM
JWE-035 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
12.3
10
uM
JWE-035 PC-3 MLTK
WISQDKEVAVKk
Lys1
12.5
10
uM
JWE-035 PC-3 PEK
DLkPSNIFFTMDDVVK
Lys2
12.6
10
uM
JWE-035 PC-3 TLK2
YVAVkIHQLNK
Lys1
12.7
10
uM
JWE-035 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
12.8
10
uM
JWE-035 PC-3 CDK10
DLkVSNLLMTDK
Lys2
12.9
10
uM
JWE-035 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
-13.1
10
uM
JWE-035 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.3
10
uM
JWE-035 PC-3 NDR2
DTGHIYAMkILR
Lys1
13.3
10
uM
JWE-035 PC-3 CDK5
DLkPQNLLINR
Lys2
13.4
10
uM
JWE-035 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-1.4
10
uM
JWE-035 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
1.4
10
uM
JWE-035 PC-3 SLK
DLkAGNILFTLDGDIK
Lys2
14.0
10
uM
JWE-035 PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
-14.2
10
uM
JWE-035 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
14.5
10
uM
JWE-035 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
14.6
10
uM
JWE-035 PC-3 CDK14
LVALkVIR
Lys1
14.6
10
uM
JWE-035 PC-3 MK11
QELNkTVWEVPQR
Other
-14.7
10
uM
JWE-035 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
14.8
10
uM
JWE-035 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
14.8
10
uM
JWE-035 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
14.8
10
uM