JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JWE-035 | HeLa | PLK1 | DLkLGNLFLNEDLEVK | Lys2 | -1.2 | 10 | uM |
JWE-035 | PC-3 | PDK1 | EYAIkILEK | Lys1 | 12.1 | 10 | uM |
JWE-035 | HeLa | TEC | YVLDDQYTSSSGAkFPVK | Activation Loop | 12.1 | 10 | uM |
JWE-035 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | 12.2 | 10 | uM |
JWE-035 | PC-3 | EphA7 | VIEDDPEAVYTTTGGkIPVR | Activation Loop | 12.3 | 10 | uM |
JWE-035 | PC-3 | MLTK | WISQDKEVAVKk | Lys1 | 12.5 | 10 | uM |
JWE-035 | PC-3 | PEK | DLkPSNIFFTMDDVVK | Lys2 | 12.6 | 10 | uM |
JWE-035 | PC-3 | TLK2 | YVAVkIHQLNK | Lys1 | 12.7 | 10 | uM |
JWE-035 | HeLa | JAK2 domain2 | IGDFGLTkVLPQDKEYYK | Activation Loop | 12.8 | 10 | uM |
JWE-035 | PC-3 | CDK10 | DLkVSNLLMTDK | Lys2 | 12.9 | 10 | uM |
JWE-035 | PC-3 | WNK4 | DLkCDNVFITGPTGSVK | Lys2 | -13.1 | 10 | uM |
JWE-035 | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -13.3 | 10 | uM |
JWE-035 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 13.3 | 10 | uM |
JWE-035 | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 13.4 | 10 | uM |
JWE-035 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -1.4 | 10 | uM |
JWE-035 | PC-3 | EPHA2 | VLEDDPEATYTTSGGkIPIR | Activation Loop | 1.4 | 10 | uM |
JWE-035 | PC-3 | SLK | DLkAGNILFTLDGDIK | Lys2 | 14.0 | 10 | uM |
JWE-035 | PC-3 | p38a | DLkPSNLAVNEDCELK | Lys2 | -14.2 | 10 | uM |
JWE-035 | HeLa | WEE1 | YIHSMSLVHMDIkPSNIFISR | Lys2 | 14.5 | 10 | uM |
JWE-035 | HeLa | FER | TSVAVkTCKEDLPQELK | Lys1 | 14.6 | 10 | uM |
JWE-035 | PC-3 | CDK14 | LVALkVIR | Lys1 | 14.6 | 10 | uM |
JWE-035 | PC-3 | MK11 | QELNkTVWEVPQR | Other | -14.7 | 10 | uM |
JWE-035 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | 14.8 | 10 | uM |
JWE-035 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | 14.8 | 10 | uM |
JWE-035 | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 14.8 | 10 | uM |