JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 PKR
DLkPSNIFLVDTK
Lys2
8.4
10
uM
JWE-035 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
8.4
10
uM
JWE-035 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
8.5
10
uM
JWE-035 HeLa LATS1
ALYATkTLR
Lys1
-8.8
10
uM
JWE-035 HeLa p38d,p38g
DLkPGNLAVNEDCELK
Lys2
-8.8
10
uM
JWE-035 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
91.1
10
uM
JWE-035 PC-3 MARK2,MARK3
DLkAENLLLDADMNIK
Lys2
9.2
10
uM
JWE-035 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
93.2
10
uM
JWE-035 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-9.4
10
uM
JWE-035 HeLa KPCI
IYAMkVVK
Lys1
9.4
10
uM
JWE-035 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
9.4
10
uM
JWE-035 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
95.4
10
uM
JWE-035 HeLa KS6B1
DLkPENIMLNHQGHVK
Lys2
9.6
10
uM
JWE-035 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
9.7
10
uM
JWE-035 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
9.8
10
uM
JWE-035 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.9
10
uM