JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
95.4
10
uM
JWE-035 PC-3 ROCK1
kLQLELNQER
Other
18.7
10
uM
JWE-035 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
10
uM
JWE-035 PC-3 MK14
QELNkTIWEVPER
Other
-5.9
10
uM
JWE-035 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
93.2
10
uM
JWE-035 PC-3 MK11
QELNkTVWEVPQR
Other
-14.7
10
uM
JWE-035 HeLa MK14
QELNkTIWEVPER
Other
7.9
10
uM
JWE-035 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
26.4
10
uM
JWE-035 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-48.5
10
uM
JWE-035 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
16.9
10
uM
JWE-035 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
8.5
10
uM
JWE-035 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.9
10
uM
JWE-035 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.3
10
uM
JWE-035 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
-401.7
10
uM
JWE-035 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
33.0
10
uM
JWE-035 HeLa PAN3
VMDPTkILITGK
5.8
10
uM