JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 SRPK1
IIHTDIkPENILLSVNEQYIR
Lys2
9.8
 10
uM
JWE-035 PC-3 SRPK1/2
FVAMkVVK
Lys1
-6.3
 10
uM
JWE-035 HeLa ULK3
EVVAIkCVAK
Lys1
8.2
 10
uM
JWE-035 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-6.9
 10
uM
JWE-035 HeLa KPCI
IYAMkVVK
Lys1
9.4
 10
uM
JWE-035 PC-3 PRP4
CNILHADIkPDNILVNESK
Lys2
-0.9
 10
uM
JWE-035 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
7.3
 10
uM
JWE-035 PC-3 CaMK2a,CaMK2b,CaMK2d,CaMK2g
DLkPENLLLASK
Lys2
-3.2
 10
uM
JWE-035 PC-3 CDK5
ETHEIVALkR
Lys1
54.2
 10
uM
JWE-035 PC-3 CK2a2
DVkPHNVMIDHQQK
Lys2
31.6
 10
uM
JWE-035 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
5.8
 10
uM
JWE-035 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
16.8
 10
uM
JWE-035 PC-3 EPHA2
EVPVAIkTLK
Lys1
8.4
 10
uM
JWE-035 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
12.3
 10
uM
JWE-035 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
22.4
 10
uM
JWE-035 HeLa GCN2
LDGCCYAVkR
Lys1
-39.6
 10
uM
JWE-035 PC-3 GCN2
LDGCCYAVkR
Lys1
18.1
 10
uM
JWE-035 HeLa JAK2 domain2
IGDFGLTkVLPQDKEYYK
Activation Loop
12.8
 10
uM
JWE-035 HeLa JAK3 domain2
IADFGLAkLLPLDKDYYVVR
Activation Loop
28.3
 10
uM
JWE-035 PC-3 M4K3
NVNTGELAAIkVIK
Lys1
18.0
 10
uM
JWE-035 PC-3 MET
DMYDKEYYSVHNkTGAK
Activation Loop
3.5
 10
uM
JWE-035 PC-3 MRCKb
DIkPDNVLLDVNGHIR
Lys2
4.7
 10
uM
JWE-035 PC-3 MK11
QELNkTVWEVPQR
Other
-14.7
 10
uM
JWE-035 PC-3 PDK1
EYAIkILEK
Lys1
12.1
 10
uM
JWE-035 PC-3 PI42C
ELPTLkDMDFLNK
ATP
78.9
 10
uM