JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 HeLa PKD2
DVAVkVIDK
Lys1
-31.1
 10
uM
JWE-035 PC-3 PKD2
DVAVkVIDK
Lys1
60.9
 10
uM
JWE-035 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
2.0
 10
uM
JWE-035 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-9.4
 10
uM
JWE-035 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
9.4
 10
uM
JWE-035 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
24.5
 10
uM
JWE-035 HeLa SYK
ISDFGLSkALR
Activation Loop
-0.1
 10
uM
JWE-035 HeLa TLK1
YAAVkIHQLNK
Lys1
-48.4
 10
uM
JWE-035 PC-3 TLK1
YAAVkIHQLNK
Lys1
37.8
 10
uM
JWE-035 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
22.8
 10
uM
JWE-035 HeLa AurB
SHFIVALkVLFK
Lys1
80.4
 10
uM
JWE-035 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
20.4
 10
uM
JWE-035 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
33.0
 10
uM
JWE-035 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-4.9
 10
uM
JWE-035 PC-3 SNRK
DLkPENVVFFEK
Lys2
5.9
 10
uM
JWE-035 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
12.1
 10
uM