JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
3.2
10
uM
JWE-035 HeLa PKD1,PKD2
NIVHCDLkPENVLLASADPFPQVK
Lys2
34.5
10
uM
JWE-035 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-6.1
10
uM
JWE-035 HeLa CaMK2g
TSTQEYAAkIINTK
Lys1
19.9
10
uM
JWE-035 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
6.6
10
uM
JWE-035 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
93.2
10
uM
JWE-035 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
14.8
10
uM
JWE-035 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
-10.2
10
uM
JWE-035 HeLa JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-3.2
10
uM
JWE-035 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
29.7
10
uM
JWE-035 HeLa SGK3
FYAVkVLQK
Lys1
4.8
10
uM
JWE-035 HeLa LATS1
ALYATkTLR
Lys1
-8.8
10
uM
JWE-035 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-1.4
10
uM
JWE-035 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-9.9
10
uM
JWE-035 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
30.5
10
uM
JWE-035 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
6.2
10
uM
JWE-035 HeLa LOK
NKETGALAAAkVIETK
Lys1
45.6
10
uM
JWE-035 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
63.0
10
uM
JWE-035 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
2.5
10
uM
JWE-035 HeLa MAP3K5,MAP3K6,MAP3K7
IAIkEIPERDSR
Lys1
-2.7
10
uM
JWE-035 HeLa MAP2K3
DVkPSNVLINK
Lys2
-1.6
10
uM
JWE-035 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
4.2
10
uM
JWE-035 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
6.7
10
uM
JWE-035 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
28.7
10
uM
JWE-035 HeLa MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
39.4
10
uM