JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
JWE-035 | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 3.2 | 10 | uM |
JWE-035 | HeLa | PKD1,PKD2 | NIVHCDLkPENVLLASADPFPQVK | Lys2 | 34.5 | 10 | uM |
JWE-035 | HeLa | IRAK4 | DIkSANILLDEAFTAK | Lys2 | -6.1 | 10 | uM |
JWE-035 | HeLa | CaMK2g | TSTQEYAAkIINTK | Lys1 | 19.9 | 10 | uM |
JWE-035 | HeLa | IRE1 | DLkPHNILISMPNAHGK | Lys2 | 6.6 | 10 | uM |
JWE-035 | HeLa | JAK1 | QLASALSYLEDKDLVHGNVCTkNLLLAR | Other | 93.2 | 10 | uM |
JWE-035 | HeLa | JAK1_domain2 | YDPEGDNTGEQVAVkSLKPESGGNHIADLKK | Lys1 | 14.8 | 10 | uM |
JWE-035 | HeLa | JAK1_domain2 | IGDFGLTkAIETDKEYYTVK | Activation Loop | -10.2 | 10 | uM |
JWE-035 | HeLa | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | -3.2 | 10 | uM |
JWE-035 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 29.7 | 10 | uM |
JWE-035 | HeLa | SGK3 | FYAVkVLQK | Lys1 | 4.8 | 10 | uM |
JWE-035 | HeLa | LATS1 | ALYATkTLR | Lys1 | -8.8 | 10 | uM |
JWE-035 | HeLa | LKB1 | DIkPGNLLLTTGGTLK | Lys2 | -1.4 | 10 | uM |
JWE-035 | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -9.9 | 10 | uM |
JWE-035 | HeLa | LOK | DLkAGNVLMTLEGDIR | Lys2 | 30.5 | 10 | uM |
JWE-035 | HeLa | ARAF | DLkSNNIFLHEGLTVK | Lys2 | 6.2 | 10 | uM |
JWE-035 | HeLa | LOK | NKETGALAAAkVIETK | Lys1 | 45.6 | 10 | uM |
JWE-035 | HeLa | AMPKa1,AMPKa2 | DLkPENVLLDAHMNAK | Lys2 | 63.0 | 10 | uM |
JWE-035 | HeLa | MAP2K1,MAP2K2 | DVkPSNILVNSR | Lys2 | 2.5 | 10 | uM |
JWE-035 | HeLa | MAP3K5,MAP3K6,MAP3K7 | IAIkEIPERDSR | Lys1 | -2.7 | 10 | uM |
JWE-035 | HeLa | MAP2K3 | DVkPSNVLINK | Lys2 | -1.6 | 10 | uM |
JWE-035 | HeLa | MK03 | DLkPSNLLINTTCDLK | Lys2 | 4.2 | 10 | uM |
JWE-035 | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 6.7 | 10 | uM |
JWE-035 | HeLa | TBK1 | TGDLFAIkVFNNISFLRPVDVQMR | Lys1 | 28.7 | 10 | uM |
JWE-035 | HeLa | MPSK1 | DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR | Lys2 | 39.4 | 10 | uM |