JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

 Full screen view
Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 ILK
WQGNDIVVkVLK
Lys1
3.0
 10
uM
JWE-035 PC-3 IRAK1
AIQFLHQDSPSLIHGDIkSSNVLLDER
Lys2
19.9
 10
uM
JWE-035 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-6.1
 10
uM
JWE-035 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
5.0
 10
uM
JWE-035 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
6.6
 10
uM
JWE-035 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
93.2
 10
uM
JWE-035 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
14.8
 10
uM
JWE-035 HeLa JAK1_domain2
IGDFGLTkAIETDKEYYTVK
Activation Loop
-10.2
 10
uM
JWE-035 HeLa JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
-3.2
 10
uM
JWE-035 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
8.4
 10
uM
JWE-035 PC-3 KHS1
NVHTGELAAVkIIK
Lys1
5.5
 10
uM
JWE-035 HeLa LATS1
ALYATkTLR
Lys1
-8.8
 10
uM
JWE-035 HeLa LKB1
DIkPGNLLLTTGGTLK
Lys2
-1.4
 10
uM
JWE-035 PC-3 LKB1
DIkPGNLLLTTGGTLK
Lys2
9.7
 10
uM
JWE-035 HeLa LOK
DLkAGNVLMTLEGDIR
Lys2
30.5
 10
uM
JWE-035 PC-3 LOK
DLkAGNVLMTLEGDIR
Lys2
16.0
 10
uM
JWE-035 HeLa LOK
NKETGALAAAkVIETK
Lys1
45.6
 10
uM
JWE-035 PC-3 LOK
NKETGALAAAkVIETK
Lys1
47.7
 10
uM
JWE-035 HeLa MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
2.5
 10
uM
JWE-035 PC-3 MAP2K1,MAP2K2
DVkPSNILVNSR
Lys2
-4.3
 10
uM
JWE-035 HeLa MAP2K3
DVkPSNVLINK
Lys2
-1.6
 10
uM
JWE-035 PC-3 MAP2K3
DVkPSNVLINK
Lys2
7.9
 10
uM
JWE-035 PC-3 MAP2K4
MVHKPSGQIMAVkR
Lys1
-3.7
 10
uM
JWE-035 PC-3 MAP2K4
DIkPSNILLDR
Lys2
-0.3
 10
uM
JWE-035 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
91.1
 10
uM