JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 PI42C
ELPTLkDMDFLNK
ATP
78.9
 10
uM
JWE-035 PC-3 EGFR
IPVAIkELR
Lys1
7.8
 10
uM
JWE-035 PC-3 RON
IQCAIkSLSR
Lys1
7.7
 10
uM
JWE-035 PC-3 PI42C
TLVIkEVSSEDIADMHSNLSNYHQYIVK
ATP
76.9
 10
uM
JWE-035 PC-3 AMPKa1,AMPKa2
VAVkILNR
Lys1
75.7
 10
uM
JWE-035 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
75.6
 10
uM
JWE-035 PC-3 ANPb
GMAFLHNSIISSHGSLkSSNCVVDSR
Lys2
7.3
 10
uM
JWE-035 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
7.3
 10
uM
JWE-035 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
7.2
 10
uM
JWE-035 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
71.7
 10
uM
JWE-035 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.1
 10
uM
JWE-035 PC-3 EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
-6.9
 10
uM
JWE-035 PC-3 MPSK1
DLkPTNILLGDEGQPVLMDLGSMNQACIHVEGSR
Lys2
68.1
 10
uM
JWE-035 PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
6.8
 10
uM
JWE-035 HeLa CDK2
DLkPQNLLINTEGAIK
Lys2
6.7
 10
uM
JWE-035 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
66.4
 10
uM
JWE-035 HeLa IRE1
DLkPHNILISMPNAHGK
Lys2
6.6
 10
uM
JWE-035 HeLa PCTAIRE2
DLkPQNLLINEK
Lys2
-6.6
 10
uM
JWE-035 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
6.5
 10
uM
JWE-035 HeLa AMPKa1,AMPKa2
DLkPENVLLDAHMNAK
Lys2
63.0
 10
uM
JWE-035 PC-3 SRPK1/2
FVAMkVVK
Lys1
-6.3
 10
uM
JWE-035 HeLa ARAF
DLkSNNIFLHEGLTVK
Lys2
6.2
 10
uM
JWE-035 HeLa MAST2,MAST4
DLkPDNLLVTSMGHIK
Lys2
6.1
 10
uM
JWE-035 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-6.1
 10
uM
JWE-035 HeLa IRAK4
DIkSANILLDEAFTAK
Lys2
-6.1
 10
uM