JWE-035 KiNativ -- single dose experiment - Dataset (ID:20100)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
JWE-035 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-6.1
 10
uM
JWE-035 PC-3 CaMK2g
TSTQEYAAkIINTK
Lys1
21.0
 10
uM
JWE-035 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
66.4
 10
uM
JWE-035 PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
16.0
 10
uM
JWE-035 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
4.9
 10
uM
JWE-035 PC-3 CDK10
DLkVSNLLMTDK
Lys2
12.9
 10
uM
JWE-035 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-13.3
 10
uM
JWE-035 PC-3 EGFR
IPVAIkELR
Lys1
7.8
 10
uM
JWE-035 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
1.4
 10
uM
JWE-035 PC-3 IRAK4
DIkSANILLDEAFTAK
Lys2
5.0
 10
uM
JWE-035 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
2.9
 10
uM
JWE-035 PC-3 CDK2
DLkPQNLLINTEGAIK
Lys2
14.8
 10
uM
JWE-035 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
34.0
 10
uM
JWE-035 PC-3 CDK5
NRETHEIVALkR
Lys1
34.0
 10
uM
JWE-035 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
-8.1
 10
uM
JWE-035 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
41.6
 10
uM
JWE-035 PC-3 ATR
FYIMMCkPK
ATP
3.6
 10
uM
JWE-035 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
7.1
 10
uM
JWE-035 PC-3 CDK9
DMkAANVLITR
Lys2
4.2
 10
uM
JWE-035 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
7.2
 10
uM
JWE-035 PC-3 CHK2
VAIkIISK
Lys1
42.7
 10
uM
JWE-035 PC-3 KC1A
DIkPDNFLMGIGR
Lys2
-0.4
 10
uM
JWE-035 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
29.0
 10
uM
JWE-035 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
8.5
 10
uM
JWE-035 PC-3 MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
17.1
 10
uM