XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
61.5
10
uM
XMD16-144 HeLa MLTK
WISQDKEVAVKk
Lys1
17.0
10
uM
XMD16-144 PC-3 MLTK
WISQDKEVAVKk
Lys1
26.2
10
uM
XMD16-144 PC-3 ILK
WQGIVVkVLK
Lys1
3.0
10
uM
XMD16-144 HeLa ILK
WQGIVVkVLK
Lys1
1.0
10
uM
XMD16-144 HeLa TLK1
YAAVkIHQLNK
Lys1
14.3
10
uM
XMD16-144 PC-3 TLK1
YAAVkIHQLNK
Lys1
-10.1
10
uM
XMD16-144 HeLa JAK1_domain2
YDPEGDNTGEQVAVkSLKPESGGNHIADLKK
Lys1
-158.2
10
uM
XMD16-144 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
10
uM
XMD16-144 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
0.2
10
uM
XMD16-144 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-3.6
10
uM
XMD16-144 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
4.4
10
uM
XMD16-144 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-13.2
10
uM
XMD16-144 HeLa STLK5
YSVkVLPWLSPEVLQQNLQGYDAK
Activation Loop
10
uM
XMD16-144 PC-3 TLK2
YVAVkIHQLNK
Lys1
9.6
10
uM
XMD16-144 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
27.3
10
uM