XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 PC-3 TAOK2
DVkAGNILLSEPGLVK
Lys2
89.8
10
uM
XMD16-144 HeLa TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
10
uM
XMD16-144 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
27.3
10
uM
XMD16-144 HeLa TLK1
YAAVkIHQLNK
Lys1
14.3
10
uM
XMD16-144 PC-3 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
4.4
10
uM
XMD16-144 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-13.2
10
uM
XMD16-144 PC-3 TLK1
YAAVkIHQLNK
Lys1
-10.1
10
uM
XMD16-144 PC-3 TLK2
YVAVkIHQLNK
Lys1
9.6
10
uM
XMD16-144 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-15.7
10
uM
XMD16-144 HeLa ULK3
EVVAIkCVAK
Lys1
14.9
10
uM
XMD16-144 HeLa WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
10
uM
XMD16-144 HeLa Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
6.7
10
uM
XMD16-144 PC-3 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
19.4
10
uM
XMD16-144 PC-3 WNK4
DLkCDNVFITGPTGSVK
Lys2
9.8
10
uM
XMD16-144 PC-3 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
6.9
10
uM
XMD16-144 HeLa ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
11.0
10
uM