XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
---|---|---|---|---|---|---|---|
XMD16-144 | HeLa | RSK1,RSK2_domain1 | DLkPENILLDEEGHIKLTDFGLSK | Lys2 | 12.1 | 10 | uM |
XMD16-144 | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | -12.3 | 10 | uM |
XMD16-144 | PC-3 | NEK6,NEK7 | DIkPANVFITATGVVK | Lys2 | -12.5 | 10 | uM |
XMD16-144 | PC-3 | NDR2 | DTGHIYAMkILR | Lys1 | 12.7 | 10 | uM |
XMD16-144 | HeLa | PAN3 | VMDPTkILITGK | -12.8 | 10 | uM | |
XMD16-144 | PC-3 | MAP3K4 | DIkGANIFLTSSGLIK | Lys2 | -12.8 | 10 | uM |
XMD16-144 | PC-3 | MAP2K6 | HVPSGQIMAVkR | Lys1 | -12.9 | 10 | uM |
XMD16-144 | PC-3 | JNK1,JNK2,JNK3 | DLkPSNIVVK | Lys2 | 12.9 | 10 | uM |
XMD16-144 | HeLa | IKKE,TBK1 | DIkPGNIMR | Lys2 | -1.3 | 10 | uM |
XMD16-144 | HeLa | TLK1 | YLNEIKPPIIHYDLkPGNILLVDGTACGEIK | Lys2 | -13.2 | 10 | uM |
XMD16-144 | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 13.9 | 10 | uM |
XMD16-144 | HeLa | PIK3CG | KkPLWLEFK | ATP | 14.3 | 10 | uM |
XMD16-144 | HeLa | TLK1 | YAAVkIHQLNK | Lys1 | 14.3 | 10 | uM |
XMD16-144 | HeLa | LYN | VAVkTLKPGTMSVQAFLEEANLMK | Lys1 | 14.3 | 10 | uM |
XMD16-144 | HeLa | KSR1,KSR2 | SkNVFYDNGK | Protein Kinase Domain | -14.4 | 10 | uM |
XMD16-144 | HeLa | SYK | ISDFGLSkALR | Activation Loop | 14.5 | 10 | uM |
XMD16-144 | PC-3 | MK03 | DLkPSNLLINTTCDLK | Lys2 | 14.5 | 10 | uM |
XMD16-144 | HeLa | MLK3 | DLkSNNILLLQPIESDDMEHK | Lys2 | -14.6 | 10 | uM |
XMD16-144 | PC-3 | p38d,p38g | DLkPGNLAVNEDCELK | Lys2 | 14.6 | 10 | uM |
XMD16-144 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | 14.6 | 10 | uM |
XMD16-144 | PC-3 | MAST3 | DLkPDNLLITSLGHIK | Lys2 | 14.7 | 10 | uM |
XMD16-144 | HeLa | ULK3 | EVVAIkCVAK | Lys1 | 14.9 | 10 | uM |
XMD16-144 | HeLa | NEK9 | LGDYGLAkK | Activation Loop | 1.5 | 10 | uM |
XMD16-144 | PC-3 | PHKg2 | ATGHEFAVkIMEVTAER | Lys1 | -15.1 | 10 | uM |
XMD16-144 | HeLa | ULK1 | DLkPQNILLSNPAGR | Lys2 | -15.7 | 10 | uM |