XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
12.1
10
uM
XMD16-144 PC-3 CK1d,CK1e
DVkPDNFLMGLGKK
Lys2
-12.3
10
uM
XMD16-144 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-12.5
10
uM
XMD16-144 PC-3 NDR2
DTGHIYAMkILR
Lys1
12.7
10
uM
XMD16-144 HeLa PAN3
VMDPTkILITGK
-12.8
10
uM
XMD16-144 PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
-12.8
10
uM
XMD16-144 PC-3 MAP2K6
HVPSGQIMAVkR
Lys1
-12.9
10
uM
XMD16-144 PC-3 JNK1,JNK2,JNK3
DLkPSNIVVK
Lys2
12.9
10
uM
XMD16-144 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-1.3
10
uM
XMD16-144 HeLa TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
-13.2
10
uM
XMD16-144 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
13.9
10
uM
XMD16-144 HeLa PIK3CG
KkPLWLEFK
ATP
14.3
10
uM
XMD16-144 HeLa TLK1
YAAVkIHQLNK
Lys1
14.3
10
uM
XMD16-144 HeLa LYN
VAVkTLKPGTMSVQAFLEEANLMK
Lys1
14.3
10
uM
XMD16-144 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-14.4
10
uM
XMD16-144 HeLa SYK
ISDFGLSkALR
Activation Loop
14.5
10
uM
XMD16-144 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
14.5
10
uM
XMD16-144 HeLa MLK3
DLkSNNILLLQPIESDDMEHK
Lys2
-14.6
10
uM
XMD16-144 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
14.6
10
uM
XMD16-144 HeLa SMG1
DTVTIHSVGGTITILPTkTKPK
ATP
14.6
10
uM
XMD16-144 PC-3 MAST3
DLkPDNLLITSLGHIK
Lys2
14.7
10
uM
XMD16-144 HeLa ULK3
EVVAIkCVAK
Lys1
14.9
10
uM
XMD16-144 HeLa NEK9
LGDYGLAkK
Activation Loop
1.5
10
uM
XMD16-144 PC-3 PHKg2
ATGHEFAVkIMEVTAER
Lys1
-15.1
10
uM
XMD16-144 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-15.7
10
uM