XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD16-144 | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 82.5 | 10 | uM |
| XMD16-144 | PC-3 | AGK | ATVFLNPAACkGK | ATP | -17.8 | 10 | uM |
| XMD16-144 | HeLa | PIK3CG | KkPLWLEFK | ATP | 14.3 | 10 | uM |
| XMD16-144 | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 46.1 | 10 | uM |
| XMD16-144 | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 73.5 | 10 | uM |
| XMD16-144 | HeLa | SMG1 | DTVTIHSVGGTITILPTkTKPK | ATP | 14.6 | 10 | uM |
| XMD16-144 | PC-3 | ATR | FYIMMCkPK | ATP | -16.0 | 10 | uM |
| XMD16-144 | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | -1.7 | 10 | uM |
| XMD16-144 | HeLa | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 73.4 | 10 | uM |
| XMD16-144 | HeLa | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 17.2 | 10 | uM |
| XMD16-144 | HeLa | PIK3C3 | TEDGGKYPVIFkHGDDLR | ATP | 36.3 | 10 | uM |
| XMD16-144 | HeLa | ATR | FYIMMCkPK | ATP | -22.3 | 10 | uM |
| XMD16-144 | PC-3 | PI42C | TLVIkEVSSEDIADMHSNLSNYHQYIVK | ATP | 84.2 | 10 | uM |
| XMD16-144 | PC-3 | PIK3CB | VFGEDSVGVIFkNGDDLRQDMLTLQMLR | ATP | 85.2 | 10 | uM |
| XMD16-144 | PC-3 | PI4KA,PI4KAP2 | SGTPMQSAAkAPYLAK | ATP | 10.8 | 10 | uM |
| XMD16-144 | HeLa | PI4KB | VPHTQAVVLNSkDK | ATP | -6.6 | 10 | uM |
| XMD16-144 | PC-3 | PI4KB | VPHTQAVVLNSkDK | ATP | 15.9 | 10 | uM |
| XMD16-144 | HeLa | RSK1,RSK4 domain1 | VLGQGSFGkVFLVR | ATP Loop | 10.2 | 10 | uM |
| XMD16-144 | HeLa | PRPK | FLSGLELVkQGAEAR | ATP Loop | 1.8 | 10 | uM |
| XMD16-144 | PC-3 | p70S6K,p70S6Kb | GGYGkVFQVR | ATP Loop | -3.3 | 10 | uM |
| XMD16-144 | HeLa | MAPKAPK3 | KYAVTDDYQLSkQVLGLGVNGK | ATP Loop | 11.8 | 10 | uM |
| XMD16-144 | HeLa | MSK1,MSK2_domain1 | VLGTGAYGkVFLVR | ATP Loop | -2.0 | 10 | uM |
| XMD16-144 | PC-3 | PRPK | FLSGLELVkQGAEAR | ATP Loop | -11.8 | 10 | uM |
| XMD16-144 | PC-3 | CASK | ETGQQFAVkIVDVAK | Lys1 | 26.8 | 10 | uM |
| XMD16-144 | PC-3 | CaMK2g | TSTQEYAAkIINTK | Lys1 | 47.3 | 10 | uM |