XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 HeLa MST3
DIkAANVLLSEHGEVK
Lys2
7.9
10
uM
XMD16-144 HeLa JAK1
QLASALSYLEDKDLVHGNVCTkNLLLAR
Other
91.0
10
uM
XMD16-144 PC-3 MK11
QELNkTVWEVPQR
Other
4.7
10
uM
XMD16-144 PC-3 MRCKb
NHHVHLYPWSSLDGAEGSFDIkLPETK
Other
-22.5
10
uM
XMD16-144 PC-3 ROCK1
kLQLELNQER
Other
3.5
10
uM
XMD16-144 HeLa MK14
QELNkTIWEVPER
Other
4.0
10
uM
XMD16-144 PC-3 MK14
QELNkTIWEVPER
Other
-30.0
10
uM
XMD16-144 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
19.2
10
uM
XMD16-144 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
0.2
10
uM
XMD16-144 HeLa KSR1,KSR2
SkNVFYDNGK
Protein Kinase Domain
-14.4
10
uM
XMD16-144 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-3.6
10
uM
XMD16-144 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
0.0
10
uM
XMD16-144 HeLa RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
18.0
10
uM
XMD16-144 PC-3 RSK2_domain2
SkRDPTEEIEILLR
Protein Kinase Domain
54.3
10
uM
XMD16-144 HeLa RSKL1_domain1
VLGVIDkVLLVMDTR
Protein Kinase Domain
9.2
10
uM
XMD16-144 HeLa PAN3
VMDPTkILITGK
-12.8
10
uM