XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 HeLa RIPK3
DLkPSNVLLDPELHVK
Lys2
-3.7
10
uM
XMD16-144 HeLa RSK1 domain1
LTDFGLSkEAIDHEK
Activation Loop
-4.7
10
uM
XMD16-144 HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
10.2
10
uM
XMD16-144 PC-3 SLK
ETSVLAAAkVIDTK
Lys1
33.2
10
uM
XMD16-144 HeLa SYK
ISDFGLSkALR
Activation Loop
14.5
10
uM
XMD16-144 HeLa TLK1
YAAVkIHQLNK
Lys1
14.3
10
uM
XMD16-144 PC-3 TLK1
YAAVkIHQLNK
Lys1
-10.1
10
uM
XMD16-144 HeLa ULK1
DLkPQNILLSNPAGR
Lys2
-15.7
10
uM
XMD16-144 HeLa AurB
SHFIVALkVLFK
Lys1
97.3
10
uM
XMD16-144 PC-3 CLK2
LTHTDLkPENILFVNSDYELTYNLEK
Lys2
10.0
10
uM
XMD16-144 HeLa IRAK3
SHLEHQSCTINMTSSSSkHLWYMPEEYIR
Protein Kinase Domain
19.2
10
uM
XMD16-144 HeLa MYO3A,MYO3B
DVkGNNILLTTEGGVK
Lys2
-7.1
10
uM
XMD16-144 PC-3 SNRK
DLkPENVVFFEK
Lys2
-8.0
10
uM
XMD16-144 HeLa TEC
YVLDDQYTSSSGAkFPVK
Activation Loop
27.3
10
uM
XMD16-144 HeLa ILK
WQGIVVkVLK
Lys1
1.0
10
uM
XMD16-144 PC-3 ILK
WQGIVVkVLK
Lys1
3.0
10
uM