XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

Filter results: >>>>
Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 PC-3 EGFR
ITDFGLAkLLGAEEK
Activation Loop
-7.5
10
uM
XMD16-144 PC-3 EphA1
LLDDFDGTYETQGGkIPIR
Activation Loop
41.9
10
uM
XMD16-144 PC-3 NEK6,NEK7
DIkPANVFITATGVVK
Lys2
-12.5
10
uM
XMD16-144 PC-3 NEK8
DLkTQNILLDK
Lys2
-28.0
10
uM
XMD16-144 PC-3 EPHA2
EVPVAIkTLK
Lys1
27.8
10
uM
XMD16-144 PC-3 NEK9
DIkTLNIFLTK
Lys2
-6.2
10
uM
XMD16-144 PC-3 EphA7
VIEDDPEAVYTTTGGkIPVR
Activation Loop
11.1
10
uM
XMD16-144 PC-3 NEK9
LGDYGLAkK
Activation Loop
8.6
10
uM
XMD16-144 PC-3 EPHB2
FLEDDTSDPTYTSALGGkIPIR
Activation Loop
43.9
10
uM
XMD16-144 PC-3 p38d,p38g
DLkPGNLAVNEDCELK
Lys2
14.6
10
uM
XMD16-144 PC-3 TLK1
YAAVkIHQLNK
Lys1
-10.1
10
uM
XMD16-144 PC-3 KS6B1
DLkPENIMLNHQGHVK
Lys2
-16.9
10
uM
XMD16-144 PC-3 p70S6K,p70S6Kb
GGYGkVFQVR
ATP Loop
-3.3
10
uM
XMD16-144 PC-3 M3K2
VYLCYDVDTGRELAVkQVQFDPDSPETSKEVNALECEIQLLK
Lys1
61.5
10
uM
XMD16-144 PC-3 CDK16
LTDNLVALkEIR
Lys1
4.2
10
uM
XMD16-144 PC-3 GCN2
LDGCCYAVkR
Lys1
3.3
10
uM