XMD16-144 KiNativ -- single dose experiment - Dataset (ID:20099)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD16-144 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-2.0
10
uM
XMD16-144 PC-3 CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
13.9
10
uM
XMD16-144 HeLa DMPK
DIkPDNILLDR
Lys2
-6.6
10
uM
XMD16-144 PC-3 DNAPK
kGGSWIQEINVAEK
ATP
82.5
10
uM
XMD16-144 HeLa DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
46.1
10
uM
XMD16-144 PC-3 DNAPK
GHDEREHPFLVkGGEDLRQDQR
ATP
73.5
10
uM
XMD16-144 HeLa eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
0.2
10
uM
XMD16-144 PC-3 eEF2K
YIkYNSNSGFVR
Protein Kinase Domain
-3.6
10
uM
XMD16-144 PC-3 EGFR
IPVAIkELR
Lys1
3.7
10
uM
XMD16-144 PC-3 EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
4.4
10
uM
XMD16-144 HeLa MK03
DLkPSNLLINTTCDLK
Lys2
-11.9
10
uM
XMD16-144 PC-3 MK03
DLkPSNLLINTTCDLK
Lys2
14.5
10
uM
XMD16-144 HeLa Erk5
DLkPSNLLVNENCELK
Lys2
96.5
10
uM
XMD16-144 PC-3 FAK
CIGEGQFGDVHQGIYMSPENPALAVAIkTCK
Lys1
80.3
10
uM
XMD16-144 HeLa FER
TSVAVkTCKEDLPQELK
Lys1
28.5
10
uM
XMD16-144 PC-3 FER
TSVAVkTCKEDLPQELK
Lys1
51.1
10
uM
XMD16-144 PC-3 FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
66.9
10
uM
XMD16-144 HeLa GCK
DTVTSELAAVkIVK
Lys1
3.1
10
uM
XMD16-144 PC-3 GCN2_domain2
DLkPVNIFLDSDDHVK
Lys2
-4.6
10
uM
XMD16-144 HeLa GSK3A
DIkPQNLLVDPDTAVLK
Lys2
-3.2
10
uM
XMD16-144 PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
27.7
10
uM
XMD16-144 HeLa IKKA
DLkPENIVLQDVGGK
Lys2
2.5
10
uM
XMD16-144 HeLa IKKE,TBK1
DIkPGNIMR
Lys2
-1.3
10
uM
XMD16-144 PC-3 IKKE,TBK1
DIkPGNIMR
Lys2
27.1
10
uM
XMD16-144 PC-3 ILK
ISMADVkFSFQCPGR
Protein Kinase Domain
0.0
10
uM