XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)
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| Small Molecule | Cell Line | Protein | Sequence | Labeling Site | % Inhibition | Assay compound conc | Conc unit |
|---|---|---|---|---|---|---|---|
| XMD11-85h | PC-3 | CDK2 | DLkPQNLLINTEGAIK | Lys2 | 6.3 | 10 | uM |
| XMD11-85h | HeLa | CDK2 | DLkPQNLLINTEGAIK | Lys2 | -4.5 | 10 | uM |
| XMD11-85h | PC-3 | CDK5 | DLkPQNLLINR | Lys2 | 0.6 | 10 | uM |
| XMD11-85h | PC-3 | CDK5 | NRETHEIVALkR | Lys1 | 16.3 | 10 | uM |
| XMD11-85h | PC-3 | CDK5 | ETHEIVALkR | Lys1 | -23.0 | 10 | uM |
| XMD11-85h | HeLa | CDK7 | DLkPNNLLLDENGVLK | Lys2 | -15.7 | 10 | uM |
| XMD11-85h | PC-3 | CDK9 | DMkAANVLITR | Lys2 | 3.3 | 10 | uM |
| XMD11-85h | HeLa | CHK1 | DIkPENLLLDER | Lys2 | -11.0 | 10 | uM |
| XMD11-85h | PC-3 | CHK2 | VAIkIISK | Lys1 | 0.6 | 10 | uM |
| XMD11-85h | PC-3 | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | 3.8 | 10 | uM |
| XMD11-85h | HeLa | CHK2 | DLkPENVLLSSQEEDCLIK | Lys2 | -20.1 | 10 | uM |
| XMD11-85h | PC-3 | CK1d,CK1e | DVkPDNFLMGLGKK | Lys2 | 14.5 | 10 | uM |
| XMD11-85h | PC-3 | CK2a2 | DVkPHNVMIDHQQK | Lys2 | 55.4 | 10 | uM |
| XMD11-85h | PC-3 | CLK2 | LTHTDLkPENILFVNSDYELTYNLEK | Lys2 | -1.0 | 10 | uM |
| XMD11-85h | HeLa | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | -8.0 | 10 | uM |
| XMD11-85h | PC-3 | CSK | VSDFGLTkEASSTQDTGKLPVK | Activation Loop | 4.0 | 10 | uM |
| XMD11-85h | HeLa | DGKA | IDPVPNTHPLLVFVNPkSGGK | ATP | 60.9 | 10 | uM |
| XMD11-85h | HeLa | DMPK | DIkPDNILLDR | Lys2 | 16.5 | 10 | uM |
| XMD11-85h | PC-3 | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | 2.7 | 10 | uM |
| XMD11-85h | HeLa | DNAPK | GHDEREHPFLVkGGEDLRQDQR | ATP | -21.2 | 10 | uM |
| XMD11-85h | PC-3 | DNAPK | kGGSWIQEINVAEK | ATP | 34.1 | 10 | uM |
| XMD11-85h | PC-3 | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | 10.7 | 10 | uM |
| XMD11-85h | HeLa | eEF2K | YIkYNSNSGFVR | Protein Kinase Domain | -28.6 | 10 | uM |
| XMD11-85h | PC-3 | EGFR | ITDFGLAkLLGAEEK | Activation Loop | 11.4 | 10 | uM |
| XMD11-85h | PC-3 | EGFR | LLGAEEKEYHAEGGkVPIK | Activation Loop | 4.3 | 10 | uM |