XMD11-85h KiNativ -- single dose experiment - Dataset (ID:20098)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
XMD11-85h PC-3 KHS1
NVHTGELAAVkIIK
Lys1
-8.6
10
uM
XMD11-85h PC-3 PI4KA,PI4KAP2
SGTPMQSAAkAPYLAK
ATP
8.6
10
uM
XMD11-85h HeLa Erk5
DLkPSNLLVNENCELK
Lys2
-8.8
10
uM
XMD11-85h PC-3 MARK2
EVAVkIIDKTQLNSSSLQK
Lys1
8.8
10
uM
XMD11-85h HeLa CAMK1D
LFAVkCIPK
Lys1
-8.9
10
uM
XMD11-85h HeLa ATR
FYIMMCkPK
ATP
-8.9
10
uM
XMD11-85h HeLa RSK1,RSK4 domain1
VLGQGSFGkVFLVR
ATP Loop
9.0
10
uM
XMD11-85h HeLa MST2
ESGQVVAIkQVPVESDLQEIIK
Lys1
9.2
10
uM
XMD11-85h HeLa MAP3K1
DVkGANLLIDSTGQR
Lys2
-9.3
10
uM
XMD11-85h PC-3 GSK3B
DIkPQNLLLDPDTAVLK
Lys2
9.4
10
uM
XMD11-85h HeLa MST1
ETGQIVAIkQVPVESDLQEIIK
Lys1
9.4
10
uM
XMD11-85h HeLa ULK3
EVVAIkCVAK
Lys1
-9.6
10
uM
XMD11-85h HeLa RSK1,RSK2_domain1
DLkPENILLDEEGHIKLTDFGLSK
Lys2
9.6
10
uM
XMD11-85h PC-3 p38a
DLkPSNLAVNEDCELK
Lys2
9.8
10
uM
XMD11-85h PC-3 MAP3K4
DIkGANIFLTSSGLIK
Lys2
-9.9
10
uM
XMD11-85h PC-3 CASK
ETGQQFAVkIVDVAK
Lys1
-9.9
10
uM