Torin2 KiNativ -- single dose experiment - Dataset (ID:20095)

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Small Molecule Cell Line Protein Sequence Labeling Site % Inhibition Assay compound conc Conc unit
Torin2 HeLa ABL,ARG
LMTGDTYTAHAGAkFPIK
Activation Loop
2.7
10
uM
Torin2 HeLa JAK1 domain2
IGDFGLTkAIETDKEYYTVKDDR
Activation Loop
52.3
10
uM
Torin2 HeLa EGFR
LLGAEEKEYHAEGGkVPIK
Activation Loop
17.9
10
uM
Torin2 HeLa Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
-23.1
10
uM
Torin2 HeLa RSK2_domain1
LTDFGLSkESIDHEKK
Activation Loop
7.1
10
uM
Torin2 HeLa MAP2K3
MCDFGISGYLVDSVAkTMDAGCKPYMAPER
Activation Loop
8.4
10
uM
Torin2 HeLa RSK1_domain1
LTDFGLSkEAIDHEKK
Activation Loop
2.9
10
uM
Torin2 HeLa PKR
IGDFGLVTSLkNDGKR
Activation Loop
7.7
10
uM
Torin2 HeLa MAP2K6
MCDFGISGYLVDSVAkTIDAGCKPYMAPER
Activation Loop
20.5
10
uM
Torin2 HeLa EPHB4
FLEENSSDPTYTSSLGGkIPIR
Activation Loop
-6.8
10
uM
Torin2 HeLa NDR1,NDR2
LSDFGLCTGLkK
Activation Loop
9.9
10
uM
Torin2 HeLa FYN,SRC,YES
QGAkFPIKWTAPEAALYGR
Activation Loop
53.1
10
uM
Torin2 HeLa FER
QEDGGVYSSSGLkQIPIKWTAPEALNYGR
Activation Loop
6.5
10
uM
Torin2 HeLa MST3,MST4,YSK1
LADFGVAGQLTDTQIkR
Activation Loop
-1.0
10
uM
Torin2 HeLa CSK
VSDFGLTkEASSTQDTGKLPVK
Activation Loop
-1.4
10
uM
Torin2 HeLa EPHA2
VLEDDPEATYTTSGGkIPIR
Activation Loop
22.2
10
uM