PLX4032 KiNativ -- dose response experiment - Dataset (ID:20092)

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Small Molecule Cell Line Protein Sequence Labeling Site IC50 Conc unit
Vemurafenib A-375 TBK1
TGDLFAIkVFNNISFLRPVDVQMR
Lys1
>10
uM
Vemurafenib A-375 TLK1
YLNEIKPPIIHYDLkPGNILLVDGTACGEIK
Lys2
>10
uM
Vemurafenib A-375 TLK2
YVAVkIHQLNKNWRDEK
Lys1
>10
uM
Vemurafenib A-375 TLK2
YVAVkIHQLNK
Lys1
>10
uM
Vemurafenib A-375 ULK3
EVVAIkCVAK
Lys1
uM
Vemurafenib A-375 ULK3
NISHLDLkPQNILLSSLEKPHLK
Lys2
>10
uM
Vemurafenib A-375 VRK2
MLDVLEYIHENEYVHGDIkAANLLLGYK
Lys2
>10
uM
Vemurafenib A-375 WEE1
YIHSMSLVHMDIkPSNIFISR
Lys2
>10
uM
Vemurafenib A-375 Wnk1,Wnk2,Wnk3
DLkCDNIFITGPTGSVK
Lys2
>10
uM
Vemurafenib A-375 Wnk1,Wnk2,Wnk4
IGDLGLATLkR
Activation Loop
>10
uM
Vemurafenib A-375 WNK4
DLkCDNVFITGPTGSVK
Lys2
>10
uM
Vemurafenib A-375 YANK3
DVkPDNILLDER
Lys2
ND
uM
Vemurafenib A-375 ZC1/HGK
TGQLAAIkVMDVTEDEEEEIKLEINMLK
Lys1
~10
uM
Vemurafenib A-375 ZC1/HGK,ZC2/TNIK,ZC3/MINK
DIkGQNVLLTENAEVK
Lys2
~10
uM
Vemurafenib A-375 ZC2/TNIK
TGQLAAIkVMDVTGDEEEEIKQEINMLKK
Lys1
1.3
uM
Vemurafenib A-375 ZC2/TNIK,ZC3/MINK
VIHRDIkGQNVLLTENAEVK
Lys2
~10
uM