HKI-272 KINOMEscan - Dataset (ID:20053)

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Small Molecule Protein % Control Assay compound conc Conc unit
Neratinib KKCC1 100.0 10
uM
Neratinib KCC4 100.0 10
uM
Neratinib CAMK1G 100.0 10
uM
Neratinib PTK6 100.0 10
uM
Neratinib CAMK2B 100.0 10
uM
Neratinib KCC2D 100.0 10
uM
Neratinib ABL1(E255K)-phosphorylated 100.0 10
uM
Neratinib ABL1(M351T)-phosphorylated 100.0 10
uM
Neratinib ABL1(F317L)-nonphosphorylated 100.0 10
uM
Neratinib AKT3 100.0 10
uM
Neratinib BRSK2 100.0 10
uM
Neratinib BRAF(V600E) 100.0 10
uM
Neratinib ANKK1 100.0 10
uM
Neratinib ALK 100.0 10
uM
Neratinib ABL1-phosphorylated 100.0 10
uM
Neratinib ABL1(H396P)-phosphorylated 100.0 10
uM
Neratinib ACVR1 100.0 10
uM
Neratinib ACVR1B 100.0 10
uM
Neratinib ACVR2A 100.0 10
uM
Neratinib ACVR2B 100.0 10
uM
Neratinib ACVRL1 100.0 10
uM
Neratinib ABL1(T315I)-phosphorylated 100.0 10
uM
Neratinib M3K5 100.0 10
uM
Neratinib CDC2L2 100.0 10
uM
Neratinib CASK 100.0 10
uM
  • Page 1 of 18
  • 1 to 25 of 442 records