HKI-272 KINOMEscan - Dataset (ID:20053)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Neratinib | KKCC1 | 100.0 | 10 | uM |
Neratinib | KCC4 | 100.0 | 10 | uM |
Neratinib | CAMK1G | 100.0 | 10 | uM |
Neratinib | PTK6 | 100.0 | 10 | uM |
Neratinib | CAMK2B | 100.0 | 10 | uM |
Neratinib | KCC2D | 100.0 | 10 | uM |
Neratinib | ABL1(E255K)-phosphorylated | 100.0 | 10 | uM |
Neratinib | ABL1(M351T)-phosphorylated | 100.0 | 10 | uM |
Neratinib | ABL1(F317L)-nonphosphorylated | 100.0 | 10 | uM |
Neratinib | AKT3 | 100.0 | 10 | uM |
Neratinib | BRSK2 | 100.0 | 10 | uM |
Neratinib | BRAF(V600E) | 100.0 | 10 | uM |
Neratinib | ANKK1 | 100.0 | 10 | uM |
Neratinib | ALK | 100.0 | 10 | uM |
Neratinib | ABL1-phosphorylated | 100.0 | 10 | uM |
Neratinib | ABL1(H396P)-phosphorylated | 100.0 | 10 | uM |
Neratinib | ACVR1 | 100.0 | 10 | uM |
Neratinib | ACVR1B | 100.0 | 10 | uM |
Neratinib | ACVR2A | 100.0 | 10 | uM |
Neratinib | ACVR2B | 100.0 | 10 | uM |
Neratinib | ACVRL1 | 100.0 | 10 | uM |
Neratinib | ABL1(T315I)-phosphorylated | 100.0 | 10 | uM |
Neratinib | M3K5 | 100.0 | 10 | uM |
Neratinib | CDC2L2 | 100.0 | 10 | uM |
Neratinib | CASK | 100.0 | 10 | uM |