GSK461364 KINOMEscan - Dataset (ID:20031)

Proteins Studied

LINCS ID Name HMS LINCS ID UniProt ID Alternative Names Provider Mutation Phosphlorylation State Domain Protein Description
200185 HCK 200185 P08631
Hemopoietic cell kinase; HCK; JTK9
KINOMEscan Wild Type; Full length
200186 HIPK1 200186 Q86Z02
Homeodomain interacting protein kinase 1; HIPK1; KIAA0630; MGC26642; MGC33446; MGC33548; Myak; Nbak2
KINOMEscan Wild Type; Partial length
200187 HIPK2 200187 Q9H2X6
Homeodomain interacting protein kinase 2; DKFZp686K02111; FLJ23711; HIPK2; PRO0593
KINOMEscan Wild Type; Partial length
200188 HIPK3 200188 Q9H422
Homeodomain interacting protein kinase 3; DYRK6; FIST3; HIPK3; PKY; YAK1
KINOMEscan Wild Type; Partial length
200189 HIPK4 200189 Q8NE63
Homeodomain interacting protein kinase 4; FLJ32818; HIPK4
KINOMEscan Wild Type; Partial length
200190 M4K1 200190 Q92918
Mitogen-activated protein kinase kinase kinase kinase 1; HPK1; MAP4K1
KINOMEscan Wild Type; Full length
200191 HUNK 200191 P57058
Hormonally up-regulated Neu-associated kinase; HUNK
KINOMEscan Wild Type; Partial length
200079 CDK5 200079 Q00535
Cyclin-dependent kinase 5; cell division protein kinase 5; PSSALRE
KINOMEscan Wild Type; Full length
200193 IGF1R 200193 P08069
Insulin-like growth factor 1 receptor; CD221; IGF1R; IGFIR; IGFR; JTK13; MGC142170; MGC142172; MGC18216
KINOMEscan Wild Type; Partial length
200194 IKKA 200194 O15111
Inhibitor of nuclear factor kappa-B kinase subunit alpha
KINOMEscan Wild Type; Full length
200195 IKKB 200195 O14920
Inhibitor of nuclear factor kappa-B kinase subunit beta
KINOMEscan Wild Type; Full length
200196 IKKE 200196 Q14164
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
KINOMEscan Wild Type; Full length
200197 INSR 200197 P06213
Insulin receptor; CD220; HHF5; INSR; IR
KINOMEscan Wild Type; Partial length
200198 INSRR 200198 P14616
Insulin receptor-related receptor; INSRR; IRR
KINOMEscan Wild Type; Partial length
200199 IRAK1 200199 P51617
Interleukin-1 receptor-associated kinase 1
KINOMEscan Wild Type; Partial length
200044 AURKA 200044 O14965
Aurora kinase A; AIK; AIRK1; ARK1; Aur2; AURA; AurA/Aur2; AURKA; AURORA2; Aurora-A; Ayk1; BTAK; IAK; IAK1; MGC34538; STK15; STK6; STK7
KINOMEscan Wild Type; Partial length
200201 IRAK4 200201 Q9NWZ3
Interleukin-1 receptor-associated kinase 4; IPD1; NY-REN-64; REN64
KINOMEscan Wild Type; Partial length
200202 ITK 200202 Q08881
IL2-inducible T-cell kinase; EMT; ITK; LYK; MGC126257; MGC126258; PSCTK2
KINOMEscan Wild Type; Partial length
200203 JAK1(JH1domain-catalytic) 200203 P23458
Janus kinase 1; JAK1; JAK1A; JAK1B; JAK1-catalytic; JTK3
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200204 JAK1(JH2domain-pseudokinase) 200204 P23458
Janus kinase 1; JAK1; JAK1~b; JAK1A; JAK1B; JAK1-pseudokinase; JTK3
KINOMEscan JH2domain-pseudokinase Wild Type; Partial length
200207 JAK2(JH1domain-catalytic) 200207 O60674
Janus kinase 2; JAK2; JAK2-catalytic; JTK10
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200209 JAK3(JH1domain-catalytic) 200209 P52333
Tyrosine-protein kinase JAK3; Janus kinase 3; JAK-3; L-JAK
KINOMEscan JH1domain-catalytic Wild Type; Partial length
200211 JNK1 200211 P45983
Mitogen-activated protein kinase 8; JNK; JNK1; JNK1A2; JNK21B1/2; MAPK8; PRKM8; SAPK1
KINOMEscan Wild Type; Full length
200147 EPHB6 200147 O15197
EPH receptor B6; EPHB6; HEP; MGC129910; MGC129911
KINOMEscan Wild Type; Partial length
200146 EPHB4 200146 P54760
Ephrin type-B receptor 4; EPHB4; HTK; MYK1; TYRO11
KINOMEscan Wild Type; Partial length