SB590885 KINOMEscan - Dataset (ID:20023)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
SB590885 | ABL2 | 55.0 | 10 | uM |
SB590885 | ABL1(Y253F)-phosphorylated | 9.1 | 10 | uM |
SB590885 | ABL1(T315I)-phosphorylated | 1.6 | 10 | uM |
SB590885 | ABL1(T315I)-nonphosphorylated | 5.4 | 10 | uM |
SB590885 | ABL1(Q252H)-phosphorylated | 3.8 | 10 | uM |
SB590885 | ABL1(Q252H)-nonphosphorylated | 3.0 | 10 | uM |
SB590885 | ABL1-phosphorylated | 6.0 | 10 | uM |
SB590885 | ABL1-nonphosphorylated | 10.0 | 10 | uM |
SB590885 | ABL1(M351T)-phosphorylated | 11.0 | 10 | uM |
SB590885 | ABL1(H396P)-phosphorylated | 6.9 | 10 | uM |
SB590885 | ABL1(H396P)-nonphosphorylated | 1.3 | 10 | uM |
SB590885 | ABL1(F317L)-phosphorylated | 37.0 | 10 | uM |
SB590885 | ABL1(F317L)-nonphosphorylated | 59.0 | 10 | uM |
SB590885 | ABL1(F317I)-phosphorylated | 81.0 | 10 | uM |
SB590885 | ABL1(F317I)-nonphosphorylated | 72.0 | 10 | uM |
SB590885 | ABL1(E255K)-phosphorylated | 8.6 | 10 | uM |
SB590885 | AAK1 | 76.0 | 10 | uM |