AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 RSK4(Kin.Dom.2-C-terminal) 17.5 10000
nM
AS-252424 PIK3C2B 19.1 10000
nM
AS-252424 EGFR(G719C) 19.2 10000
nM
AS-252424 EGFR(L858R) 20.1 10000
nM
AS-252424 RPS6KA4(Kin.Dom.2-C-terminal) 21.6 10000
nM
AS-252424 DAPK3 24.8 10000
nM
AS-252424 TIE1 25.2 10000
nM
AS-252424 PIK3CD 26.8 10000
nM
AS-252424 CLK2 27.3 10000
nM
AS-252424 EGFR(L861Q) 27.6 10000
nM
AS-252424 EGFR(G719S) 28.8 10000
nM
AS-252424 MLCK 29.1 10000
nM
AS-252424 RIPK2 31.8 10000
nM
AS-252424 TYK2(JH2domain-pseudokinase) 33.1 10000
nM
AS-252424 AAK1 35.0 10000
nM
AS-252424 RSK1(Kin.Dom.2-C-terminal) 35.1 10000
nM
AS-252424 TGFBR2 36.1 10000
nM
AS-252424 PIK3CA 38.0 10000
nM
AS-252424 JNK3 38.1 10000
nM
AS-252424 CLK4 40.3 10000
nM
AS-252424 EGFR 40.8 10000
nM
AS-252424 PIK3CA(E545K) 42.3 10000
nM
AS-252424 RPS6KA5(Kin.Dom.2-C-terminal) 43.5 10000
nM
AS-252424 BRAF(V600E) 45.6 10000
nM
AS-252424 CDK7 46.6 10000
nM