AS-252424 KINOMEscan - Dataset (ID:20341)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
AS-252424 | RSK4(Kin.Dom.2-C-terminal) | 17.5 | 10000 | nM |
AS-252424 | PIK3C2B | 19.1 | 10000 | nM |
AS-252424 | EGFR(G719C) | 19.2 | 10000 | nM |
AS-252424 | EGFR(L858R) | 20.1 | 10000 | nM |
AS-252424 | RPS6KA4(Kin.Dom.2-C-terminal) | 21.6 | 10000 | nM |
AS-252424 | DAPK3 | 24.8 | 10000 | nM |
AS-252424 | TIE1 | 25.2 | 10000 | nM |
AS-252424 | PIK3CD | 26.8 | 10000 | nM |
AS-252424 | CLK2 | 27.3 | 10000 | nM |
AS-252424 | EGFR(L861Q) | 27.6 | 10000 | nM |
AS-252424 | EGFR(G719S) | 28.8 | 10000 | nM |
AS-252424 | MLCK | 29.1 | 10000 | nM |
AS-252424 | RIPK2 | 31.8 | 10000 | nM |
AS-252424 | TYK2(JH2domain-pseudokinase) | 33.1 | 10000 | nM |
AS-252424 | AAK1 | 35.0 | 10000 | nM |
AS-252424 | RSK1(Kin.Dom.2-C-terminal) | 35.1 | 10000 | nM |
AS-252424 | TGFBR2 | 36.1 | 10000 | nM |
AS-252424 | PIK3CA | 38.0 | 10000 | nM |
AS-252424 | JNK3 | 38.1 | 10000 | nM |
AS-252424 | CLK4 | 40.3 | 10000 | nM |
AS-252424 | EGFR | 40.8 | 10000 | nM |
AS-252424 | PIK3CA(E545K) | 42.3 | 10000 | nM |
AS-252424 | RPS6KA5(Kin.Dom.2-C-terminal) | 43.5 | 10000 | nM |
AS-252424 | BRAF(V600E) | 45.6 | 10000 | nM |
AS-252424 | CDK7 | 46.6 | 10000 | nM |