AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 CIT 0.2 10000
nM
AS-252424 DRAK1 1.5 10000
nM
AS-252424 EGFR(L747-T751del,Sins) 1.9 10000
nM
AS-252424 PIM2 2.0 10000
nM
AS-252424 TIE2 2.1 10000
nM
AS-252424 PIM1 2.7 10000
nM
AS-252424 DRAK2 3.3 10000
nM
AS-252424 ERK8 3.7 10000
nM
AS-252424 PIK3CG 4.0 10000
nM
AS-252424 CSNK2A2 4.3 10000
nM
AS-252424 CSNK2A1 4.5 10000
nM
AS-252424 PIM3 4.8 10000
nM
AS-252424 HIPK1 5.0 10000
nM
AS-252424 PIK3CA(H1047R) 5.7 10000
nM
AS-252424 EGFR(L747-E749del, A750P) 5.8 10000
nM
AS-252424 TAOK1 8.5 10000
nM
AS-252424 GAK 9.3 10000
nM
AS-252424 ACVR2B 9.9 10000
nM
AS-252424 EGFR(S752-I759del) 9.9 10000
nM
AS-252424 DAPK1 10.5 10000
nM
AS-252424 BMPR2 12.5 10000
nM
AS-252424 DAPK2 12.5 10000
nM
AS-252424 EGFR(L747-S752del, P753S) 14.5 10000
nM
AS-252424 EGFR(E746-A750del) 14.6 10000
nM
AS-252424 MYLK4 17.0 10000
nM
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  • 1 to 25 of 356 records