AS-252424 KINOMEscan - Dataset (ID:20341)
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Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
AS-252424 | CIT | 0.2 | 10000 | nM |
AS-252424 | DRAK1 | 1.5 | 10000 | nM |
AS-252424 | EGFR(L747-T751del,Sins) | 1.9 | 10000 | nM |
AS-252424 | PIM2 | 2.0 | 10000 | nM |
AS-252424 | TIE2 | 2.1 | 10000 | nM |
AS-252424 | PIM1 | 2.7 | 10000 | nM |
AS-252424 | DRAK2 | 3.3 | 10000 | nM |
AS-252424 | ERK8 | 3.7 | 10000 | nM |
AS-252424 | PIK3CG | 4.0 | 10000 | nM |
AS-252424 | CSNK2A2 | 4.3 | 10000 | nM |
AS-252424 | CSNK2A1 | 4.5 | 10000 | nM |
AS-252424 | PIM3 | 4.8 | 10000 | nM |
AS-252424 | HIPK1 | 5.0 | 10000 | nM |
AS-252424 | PIK3CA(H1047R) | 5.7 | 10000 | nM |
AS-252424 | EGFR(L747-E749del, A750P) | 5.8 | 10000 | nM |
AS-252424 | TAOK1 | 8.5 | 10000 | nM |
AS-252424 | GAK | 9.3 | 10000 | nM |
AS-252424 | ACVR2B | 9.9 | 10000 | nM |
AS-252424 | EGFR(S752-I759del) | 9.9 | 10000 | nM |
AS-252424 | DAPK1 | 10.5 | 10000 | nM |
AS-252424 | BMPR2 | 12.5 | 10000 | nM |
AS-252424 | DAPK2 | 12.5 | 10000 | nM |
AS-252424 | EGFR(L747-S752del, P753S) | 14.5 | 10000 | nM |
AS-252424 | EGFR(E746-A750del) | 14.6 | 10000 | nM |
AS-252424 | MYLK4 | 17.0 | 10000 | nM |