AS-252424 KINOMEscan - Dataset (ID:20341)

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Small Molecule Protein % Control Assay compound conc Conc unit
AS-252424 KGP2 97.3 10000
nM
AS-252424 PRKR 100.0 10000
nM
AS-252424 PRKX 89.5 10000
nM
AS-252424 FAK2 100.0 10000
nM
AS-252424 RAF1 99.2 10000
nM
AS-252424 RET 100.0 10000
nM
AS-252424 RET(M918T) 85.6 10000
nM
AS-252424 RET(V804L) 90.7 10000
nM
AS-252424 RET(V804M) 100.0 10000
nM
AS-252424 RIOK1 96.6 10000
nM
AS-252424 RIOK2 100.0 10000
nM
AS-252424 RIOK3 95.5 10000
nM
AS-252424 RIPK1 95.9 10000
nM
AS-252424 RIPK2 31.8 10000
nM
AS-252424 RIPK4 100.0 10000
nM
AS-252424 ROCK2 96.2 10000
nM
AS-252424 ROS1 99.8 10000
nM
AS-252424 RPS6KA4(Kin.Dom.1-N-terminal) 90.3 10000
nM
AS-252424 RPS6KA4(Kin.Dom.2-C-terminal) 21.6 10000
nM
AS-252424 RPS6KA5(Kin.Dom.1-N-terminal) 100.0 10000
nM
AS-252424 RPS6KA5(Kin.Dom.2-C-terminal) 43.5 10000
nM
AS-252424 RSK1(Kin.Dom.1-N-terminal) 81.6 10000
nM
AS-252424 RSK1(Kin.Dom.2-C-terminal) 35.1 10000
nM
AS-252424 RSK2(Kin.Dom.1-N-terminal) 100.0 10000
nM
AS-252424 RSK3(Kin.Dom.1-N-terminal) 100.0 10000
nM