Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Palbociclib | CDK7 | 100.0 | 100 | nM |
Palbociclib | CDK7 | 100.0 | 1000 | nM |
Palbociclib | CDK8 | 100.0 | 100 | nM |
Palbociclib | CDK8 | 93.0 | 1000 | nM |
Palbociclib | CDK9 | 100.0 | 100 | nM |
Palbociclib | CDK9 | 97.0 | 1000 | nM |
Palbociclib | CDKL1 | 74.0 | 100 | nM |
Palbociclib | CDKL1 | 91.0 | 1000 | nM |
Palbociclib | CDKL2 | 95.0 | 100 | nM |
Palbociclib | CDKL2 | 71.0 | 1000 | nM |
Palbociclib | CDKL3 | 93.0 | 100 | nM |
Palbociclib | CDKL3 | 100.0 | 1000 | nM |
Palbociclib | CDKL5 | 100.0 | 100 | nM |
Palbociclib | CDKL5 | 99.0 | 1000 | nM |
Palbociclib | CHEK1 | 100.0 | 100 | nM |
Palbociclib | CHEK1 | 100.0 | 1000 | nM |
Palbociclib | CHK2 | 100.0 | 100 | nM |
Palbociclib | CHK2 | 100.0 | 1000 | nM |
Palbociclib | CIT | 100.0 | 100 | nM |
Palbociclib | CIT | 90.0 | 1000 | nM |
Palbociclib | CLK1 | 74.0 | 100 | nM |
Palbociclib | CLK1 | 10.0 | 1000 | nM |
Palbociclib | CLK2 | 76.0 | 100 | nM |
Palbociclib | CLK2 | 18.0 | 1000 | nM |
Palbociclib | CLK3 | 100.0 | 100 | nM |