Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib CDK7 100.0 100
nM
Palbociclib CDK7 100.0 1000
nM
Palbociclib CDK8 100.0 100
nM
Palbociclib CDK8 93.0 1000
nM
Palbociclib CDK9 100.0 100
nM
Palbociclib CDK9 97.0 1000
nM
Palbociclib CDKL1 74.0 100
nM
Palbociclib CDKL1 91.0 1000
nM
Palbociclib CDKL2 95.0 100
nM
Palbociclib CDKL2 71.0 1000
nM
Palbociclib CDKL3 93.0 100
nM
Palbociclib CDKL3 100.0 1000
nM
Palbociclib CDKL5 100.0 100
nM
Palbociclib CDKL5 99.0 1000
nM
Palbociclib CHEK1 100.0 100
nM
Palbociclib CHEK1 100.0 1000
nM
Palbociclib CHK2 100.0 100
nM
Palbociclib CHK2 100.0 1000
nM
Palbociclib CIT 100.0 100
nM
Palbociclib CIT 90.0 1000
nM
Palbociclib CLK1 74.0 100
nM
Palbociclib CLK1 10.0 1000
nM
Palbociclib CLK2 76.0 100
nM
Palbociclib CLK2 18.0 1000
nM
Palbociclib CLK3 100.0 100
nM