Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib TRKA 30.0 1000
nM
Palbociclib TRKB 100.0 100
nM
Palbociclib TRKB 100.0 1000
nM
Palbociclib TRKC 100.0 100
nM
Palbociclib TRKC 100.0 1000
nM
Palbociclib TRPM6 95.0 100
nM
Palbociclib TRPM6 100.0 1000
nM
Palbociclib TSSK1 100.0 100
nM
Palbociclib TSSK1 98.0 1000
nM
Palbociclib TSSK3 100.0 100
nM
Palbociclib TSSK3 100.0 1000
nM
Palbociclib TTK 64.0 100
nM
Palbociclib TTK 59.0 1000
nM
Palbociclib TXK 100.0 100
nM
Palbociclib TXK 100.0 1000
nM
Palbociclib TYK2(JH1domain-catalytic) 100.0 100
nM
Palbociclib TYK2(JH1domain-catalytic) 100.0 1000
nM
Palbociclib TYK2(JH2domain-pseudokinase) 100.0 100
nM
Palbociclib TYK2(JH2domain-pseudokinase) 100.0 1000
nM
Palbociclib TYRO3 89.0 100
nM
Palbociclib TYRO3 96.0 1000
nM
Palbociclib ULK1 100.0 100
nM
Palbociclib ULK1 100.0 1000
nM
Palbociclib ULK2 25.0 100
nM
Palbociclib ULK2 1.4 1000
nM