Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Palbociclib | RET(V804M) | 100.0 | 100 | nM |
Palbociclib | RET(V804M) | 93.0 | 1000 | nM |
Palbociclib | RIOK1 | 71.0 | 100 | nM |
Palbociclib | RIOK1 | 58.0 | 1000 | nM |
Palbociclib | RIOK2 | 100.0 | 100 | nM |
Palbociclib | RIOK2 | 100.0 | 1000 | nM |
Palbociclib | RIOK3 | 89.0 | 100 | nM |
Palbociclib | RIOK3 | 70.0 | 1000 | nM |
Palbociclib | RIPK1 | 100.0 | 100 | nM |
Palbociclib | RIPK1 | 100.0 | 1000 | nM |
Palbociclib | RIPK2 | 100.0 | 100 | nM |
Palbociclib | RIPK2 | 96.0 | 1000 | nM |
Palbociclib | RIPK4 | 100.0 | 100 | nM |
Palbociclib | RIPK4 | 100.0 | 1000 | nM |
Palbociclib | RIPK5 | 100.0 | 100 | nM |
Palbociclib | RIPK5 | 100.0 | 1000 | nM |
Palbociclib | ROCK1 | 100.0 | 100 | nM |
Palbociclib | ROCK1 | 100.0 | 1000 | nM |
Palbociclib | ROCK2 | 100.0 | 100 | nM |
Palbociclib | ROCK2 | 100.0 | 1000 | nM |
Palbociclib | ROS1 | 99.0 | 100 | nM |
Palbociclib | ROS1 | 100.0 | 1000 | nM |
Palbociclib | RPS6KA4(Kin.Dom.1-N-terminal) | 100.0 | 100 | nM |
Palbociclib | RPS6KA4(Kin.Dom.1-N-terminal) | 100.0 | 1000 | nM |
Palbociclib | RPS6KA4(Kin.Dom.2-C-terminal) | 100.0 | 100 | nM |