Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib RET(V804M) 100.0 100
nM
Palbociclib RET(V804M) 93.0 1000
nM
Palbociclib RIOK1 71.0 100
nM
Palbociclib RIOK1 58.0 1000
nM
Palbociclib RIOK2 100.0 100
nM
Palbociclib RIOK2 100.0 1000
nM
Palbociclib RIOK3 89.0 100
nM
Palbociclib RIOK3 70.0 1000
nM
Palbociclib RIPK1 100.0 100
nM
Palbociclib RIPK1 100.0 1000
nM
Palbociclib RIPK2 100.0 100
nM
Palbociclib RIPK2 96.0 1000
nM
Palbociclib RIPK4 100.0 100
nM
Palbociclib RIPK4 100.0 1000
nM
Palbociclib RIPK5 100.0 100
nM
Palbociclib RIPK5 100.0 1000
nM
Palbociclib ROCK1 100.0 100
nM
Palbociclib ROCK1 100.0 1000
nM
Palbociclib ROCK2 100.0 100
nM
Palbociclib ROCK2 100.0 1000
nM
Palbociclib ROS1 99.0 100
nM
Palbociclib ROS1 100.0 1000
nM
Palbociclib RPS6KA4(Kin.Dom.1-N-terminal) 100.0 100
nM
Palbociclib RPS6KA4(Kin.Dom.1-N-terminal) 100.0 1000
nM
Palbociclib RPS6KA4(Kin.Dom.2-C-terminal) 100.0 100
nM