Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Palbociclib | PIK3CA(C420R) | 91.0 | 100 | nM |
| Palbociclib | PIK3CA(C420R) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(E542K) | 93.0 | 100 | nM |
| Palbociclib | PIK3CA(E542K) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(E545A) | 74.0 | 100 | nM |
| Palbociclib | PIK3CA(E545A) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(E545K) | 50.0 | 100 | nM |
| Palbociclib | PIK3CA(E545K) | 55.0 | 1000 | nM |
| Palbociclib | PIK3CA(H1047L) | 100.0 | 100 | nM |
| Palbociclib | PIK3CA(H1047L) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(H1047Y) | 86.0 | 100 | nM |
| Palbociclib | PIK3CA(H1047Y) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(I800L) | 97.0 | 100 | nM |
| Palbociclib | PIK3CA(I800L) | 80.0 | 1000 | nM |
| Palbociclib | PIK3CA(M1043I) | 96.0 | 100 | nM |
| Palbociclib | PIK3CA(M1043I) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CA(Q546K) | 100.0 | 100 | nM |
| Palbociclib | PIK3CA(Q546K) | 100.0 | 1000 | nM |
| Palbociclib | PIK3CB | 100.0 | 100 | nM |
| Palbociclib | PIK3CB | 100.0 | 1000 | nM |
| Palbociclib | PIK3CD | 100.0 | 100 | nM |
| Palbociclib | PIK3CD | 68.0 | 1000 | nM |
| Palbociclib | PIK3CG | 100.0 | 100 | nM |
| Palbociclib | PIK3CG | 93.0 | 1000 | nM |
| Palbociclib | PIK4CB | 100.0 | 100 | nM |