Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Palbociclib | AMPK-alpha2 | 100.0 | 100 | nM |
Palbociclib | EGFR(L858R,T790M) | 100.0 | 100 | nM |
Palbociclib | CAMKK2 | 100.0 | 100 | nM |
Palbociclib | EGFR(L861Q) | 95.0 | 100 | nM |
Palbociclib | AAK1 | 99.0 | 100 | nM |
Palbociclib | EGFR(S752-I759del) | 92.0 | 100 | nM |
Palbociclib | CASK | 71.0 | 100 | nM |
Palbociclib | EGFR(T790M) | 100.0 | 100 | nM |
Palbociclib | ANKK1 | 100.0 | 100 | nM |
Palbociclib | EIF2AK1 | 100.0 | 100 | nM |
Palbociclib | CDC2L1 | 100.0 | 100 | nM |
Palbociclib | EPHA1 | 86.0 | 100 | nM |
Palbociclib | ABL2 | 100.0 | 100 | nM |
Palbociclib | EPHA2 | 83.0 | 100 | nM |
Palbociclib | CDC2L2 | 100.0 | 100 | nM |
Palbociclib | EPHA3 | 100.0 | 100 | nM |
Palbociclib | NUAK1 | 100.0 | 100 | nM |
Palbociclib | EPHA4 | 100.0 | 100 | nM |
Palbociclib | CDC2L5 | 99.0 | 100 | nM |
Palbociclib | EPHA5 | 100.0 | 100 | nM |
Palbociclib | ABL1(M351T)-phosphorylated | 100.0 | 100 | nM |
Palbociclib | EPHA6 | 100.0 | 100 | nM |
Palbociclib | CDK11 | 95.0 | 100 | nM |
Palbociclib | EPHA7 | 100.0 | 100 | nM |
Palbociclib | MST2 | 100.0 | 100 | nM |