Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib AMPK-alpha2 100.0 100
nM
Palbociclib EGFR(L858R,T790M) 100.0 100
nM
Palbociclib CAMKK2 100.0 100
nM
Palbociclib EGFR(L861Q) 95.0 100
nM
Palbociclib AAK1 99.0 100
nM
Palbociclib EGFR(S752-I759del) 92.0 100
nM
Palbociclib CASK 71.0 100
nM
Palbociclib EGFR(T790M) 100.0 100
nM
Palbociclib ANKK1 100.0 100
nM
Palbociclib EIF2AK1 100.0 100
nM
Palbociclib CDC2L1 100.0 100
nM
Palbociclib EPHA1 86.0 100
nM
Palbociclib ABL2 100.0 100
nM
Palbociclib EPHA2 83.0 100
nM
Palbociclib CDC2L2 100.0 100
nM
Palbociclib EPHA3 100.0 100
nM
Palbociclib NUAK1 100.0 100
nM
Palbociclib EPHA4 100.0 100
nM
Palbociclib CDC2L5 99.0 100
nM
Palbociclib EPHA5 100.0 100
nM
Palbociclib ABL1(M351T)-phosphorylated 100.0 100
nM
Palbociclib EPHA6 100.0 100
nM
Palbociclib CDK11 95.0 100
nM
Palbociclib EPHA7 100.0 100
nM
Palbociclib MST2 100.0 100
nM