Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Palbociclib | MAST1 | 100.0 | 100 | nM |
Palbociclib | MAST1 | 87.0 | 1000 | nM |
Palbociclib | MP2K1 | 98.0 | 100 | nM |
Palbociclib | MP2K1 | 93.0 | 1000 | nM |
Palbociclib | MP2K2 | 86.0 | 100 | nM |
Palbociclib | MP2K2 | 89.0 | 1000 | nM |
Palbociclib | MP2K3 | 92.0 | 100 | nM |
Palbociclib | MP2K3 | 87.0 | 1000 | nM |
Palbociclib | MP2K4 | 100.0 | 100 | nM |
Palbociclib | MP2K4 | 100.0 | 1000 | nM |
Palbociclib | MP2K5 | 83.0 | 100 | nM |
Palbociclib | MP2K5 | 94.0 | 1000 | nM |
Palbociclib | MP2K6 | 100.0 | 100 | nM |
Palbociclib | MP2K6 | 100.0 | 1000 | nM |
Palbociclib | MELK | 89.0 | 100 | nM |
Palbociclib | MELK | 84.0 | 1000 | nM |
Palbociclib | MERTK | 100.0 | 100 | nM |
Palbociclib | MERTK | 98.0 | 1000 | nM |
Palbociclib | MET | 100.0 | 100 | nM |
Palbociclib | MET | 100.0 | 1000 | nM |
Palbociclib | MET(M1250T) | 99.0 | 100 | nM |
Palbociclib | MET(M1250T) | 97.0 | 1000 | nM |
Palbociclib | MET(Y1235D) | 96.0 | 100 | nM |
Palbociclib | MET(Y1235D) | 53.0 | 1000 | nM |
Palbociclib | MINK | 92.0 | 100 | nM |