Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib MAST1 100.0 100
nM
Palbociclib MAST1 87.0 1000
nM
Palbociclib MP2K1 98.0 100
nM
Palbociclib MP2K1 93.0 1000
nM
Palbociclib MP2K2 86.0 100
nM
Palbociclib MP2K2 89.0 1000
nM
Palbociclib MP2K3 92.0 100
nM
Palbociclib MP2K3 87.0 1000
nM
Palbociclib MP2K4 100.0 100
nM
Palbociclib MP2K4 100.0 1000
nM
Palbociclib MP2K5 83.0 100
nM
Palbociclib MP2K5 94.0 1000
nM
Palbociclib MP2K6 100.0 100
nM
Palbociclib MP2K6 100.0 1000
nM
Palbociclib MELK 89.0 100
nM
Palbociclib MELK 84.0 1000
nM
Palbociclib MERTK 100.0 100
nM
Palbociclib MERTK 98.0 1000
nM
Palbociclib MET 100.0 100
nM
Palbociclib MET 100.0 1000
nM
Palbociclib MET(M1250T) 99.0 100
nM
Palbociclib MET(M1250T) 97.0 1000
nM
Palbociclib MET(Y1235D) 96.0 100
nM
Palbociclib MET(Y1235D) 53.0 1000
nM
Palbociclib MINK 92.0 100
nM