Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
---|---|---|---|---|
Palbociclib | INSR | 100.0 | 100 | nM |
Palbociclib | INSR | 100.0 | 1000 | nM |
Palbociclib | INSRR | 100.0 | 100 | nM |
Palbociclib | INSRR | 100.0 | 1000 | nM |
Palbociclib | IRAK1 | 100.0 | 100 | nM |
Palbociclib | IRAK1 | 80.0 | 1000 | nM |
Palbociclib | IRAK3 | 100.0 | 100 | nM |
Palbociclib | IRAK3 | 100.0 | 1000 | nM |
Palbociclib | IRAK4 | 100.0 | 100 | nM |
Palbociclib | IRAK4 | 100.0 | 1000 | nM |
Palbociclib | ITK | 100.0 | 100 | nM |
Palbociclib | ITK | 100.0 | 1000 | nM |
Palbociclib | JAK1(JH1domain-catalytic) | 96.0 | 100 | nM |
Palbociclib | JAK1(JH1domain-catalytic) | 100.0 | 1000 | nM |
Palbociclib | JAK1(JH2domain-pseudokinase) | 86.0 | 100 | nM |
Palbociclib | JAK1(JH2domain-pseudokinase) | 85.0 | 1000 | nM |
Palbociclib | JAK2(JH1domain-catalytic) | 100.0 | 100 | nM |
Palbociclib | JAK2(JH1domain-catalytic) | 61.0 | 1000 | nM |
Palbociclib | JAK3(JH1domain-catalytic) | 94.0 | 100 | nM |
Palbociclib | JAK3(JH1domain-catalytic) | 72.0 | 1000 | nM |
Palbociclib | JNK1 | 100.0 | 100 | nM |
Palbociclib | JNK1 | 69.0 | 1000 | nM |
Palbociclib | MK09 | 100.0 | 100 | nM |
Palbociclib | MK09 | 55.0 | 1000 | nM |
Palbociclib | JNK3 | 100.0 | 100 | nM |