Palbociclib KINOMEscan - Dataset (ID:20339)

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Small Molecule Protein % Control Assay compound conc Conc unit
Palbociclib INSR 100.0 100
nM
Palbociclib INSR 100.0 1000
nM
Palbociclib INSRR 100.0 100
nM
Palbociclib INSRR 100.0 1000
nM
Palbociclib IRAK1 100.0 100
nM
Palbociclib IRAK1 80.0 1000
nM
Palbociclib IRAK3 100.0 100
nM
Palbociclib IRAK3 100.0 1000
nM
Palbociclib IRAK4 100.0 100
nM
Palbociclib IRAK4 100.0 1000
nM
Palbociclib ITK 100.0 100
nM
Palbociclib ITK 100.0 1000
nM
Palbociclib JAK1(JH1domain-catalytic) 96.0 100
nM
Palbociclib JAK1(JH1domain-catalytic) 100.0 1000
nM
Palbociclib JAK1(JH2domain-pseudokinase) 86.0 100
nM
Palbociclib JAK1(JH2domain-pseudokinase) 85.0 1000
nM
Palbociclib JAK2(JH1domain-catalytic) 100.0 100
nM
Palbociclib JAK2(JH1domain-catalytic) 61.0 1000
nM
Palbociclib JAK3(JH1domain-catalytic) 94.0 100
nM
Palbociclib JAK3(JH1domain-catalytic) 72.0 1000
nM
Palbociclib JNK1 100.0 100
nM
Palbociclib JNK1 69.0 1000
nM
Palbociclib MK09 100.0 100
nM
Palbociclib MK09 55.0 1000
nM
Palbociclib JNK3 100.0 100
nM