Palbociclib KINOMEscan - Dataset (ID:20339)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Palbociclib | FGR | 98.0 | 1000 | nM |
| Palbociclib | VGFR1 | 92.0 | 100 | nM |
| Palbociclib | VGFR1 | 98.0 | 1000 | nM |
| Palbociclib | FLT3 | 98.0 | 100 | nM |
| Palbociclib | FLT3 | 77.0 | 1000 | nM |
| Palbociclib | FLT3(D835H) | 100.0 | 100 | nM |
| Palbociclib | FLT3(D835H) | 75.0 | 1000 | nM |
| Palbociclib | FLT3(D835V) | 66.0 | 100 | nM |
| Palbociclib | FLT3(D835V) | 44.0 | 1000 | nM |
| Palbociclib | FLT3(D835Y) | 100.0 | 100 | nM |
| Palbociclib | FLT3(D835Y) | 66.0 | 1000 | nM |
| Palbociclib | FLT3(ITD) | 100.0 | 100 | nM |
| Palbociclib | FLT3(ITD) | 87.0 | 1000 | nM |
| Palbociclib | FLT3(ITD,D835V) | 83.0 | 100 | nM |
| Palbociclib | FLT3(ITD,D835V) | 24.0 | 1000 | nM |
| Palbociclib | FLT3(ITD,F691L) | 94.0 | 100 | nM |
| Palbociclib | FLT3(ITD,F691L) | 58.0 | 1000 | nM |
| Palbociclib | FLT3(K663Q) | 100.0 | 100 | nM |
| Palbociclib | FLT3(K663Q) | 100.0 | 1000 | nM |
| Palbociclib | FLT3(N841I) | 100.0 | 100 | nM |
| Palbociclib | FLT3(N841I) | 100.0 | 1000 | nM |
| Palbociclib | FLT3(R834Q) | 100.0 | 100 | nM |
| Palbociclib | FLT3(R834Q) | 100.0 | 1000 | nM |
| Palbociclib | FLT3-autoinhibited | 100.0 | 100 | nM |
| Palbociclib | FLT3-autoinhibited | 100.0 | 1000 | nM |