Abemaciclib KINOMEscan - Dataset (ID:20338)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Abemaciclib | INSR | 100.0 | 100 | nM |
| Abemaciclib | INSR | 99.0 | 1000 | nM |
| Abemaciclib | INSRR | 100.0 | 100 | nM |
| Abemaciclib | INSRR | 97.0 | 1000 | nM |
| Abemaciclib | IRAK1 | 0.9 | 100 | nM |
| Abemaciclib | IRAK1 | 0.2 | 1000 | nM |
| Abemaciclib | IRAK3 | 89.0 | 100 | nM |
| Abemaciclib | IRAK3 | 46.0 | 1000 | nM |
| Abemaciclib | IRAK4 | 100.0 | 100 | nM |
| Abemaciclib | IRAK4 | 99.0 | 1000 | nM |
| Abemaciclib | ITK | 97.0 | 100 | nM |
| Abemaciclib | ITK | 97.0 | 1000 | nM |
| Abemaciclib | JAK1(JH1domain-catalytic) | 100.0 | 100 | nM |
| Abemaciclib | JAK1(JH1domain-catalytic) | 100.0 | 1000 | nM |
| Abemaciclib | JAK1(JH2domain-pseudokinase) | 99.0 | 100 | nM |
| Abemaciclib | JAK1(JH2domain-pseudokinase) | 90.0 | 1000 | nM |
| Abemaciclib | JAK2(JH1domain-catalytic) | 83.0 | 100 | nM |
| Abemaciclib | JAK2(JH1domain-catalytic) | 50.0 | 1000 | nM |
| Abemaciclib | JAK3(JH1domain-catalytic) | 49.0 | 100 | nM |
| Abemaciclib | JAK3(JH1domain-catalytic) | 1.8 | 1000 | nM |
| Abemaciclib | JNK1 | 42.0 | 100 | nM |
| Abemaciclib | JNK1 | 4.0 | 1000 | nM |
| Abemaciclib | MK09 | 90.0 | 100 | nM |
| Abemaciclib | MK09 | 21.0 | 1000 | nM |
| Abemaciclib | JNK3 | 60.0 | 100 | nM |