Abemaciclib KINOMEscan - Dataset (ID:20338)
Download: Excel (XLSX), Comma-separated (CSV)
| Small Molecule | Protein | % Control | Assay compound conc | Conc unit |
|---|---|---|---|---|
| Abemaciclib | FGR | 93.0 | 1000 | nM |
| Abemaciclib | VGFR1 | 95.0 | 100 | nM |
| Abemaciclib | VGFR1 | 87.0 | 1000 | nM |
| Abemaciclib | FLT3 | 85.0 | 100 | nM |
| Abemaciclib | FLT3 | 69.0 | 1000 | nM |
| Abemaciclib | FLT3(D835H) | 78.0 | 100 | nM |
| Abemaciclib | FLT3(D835H) | 39.0 | 1000 | nM |
| Abemaciclib | FLT3(D835V) | 20.0 | 100 | nM |
| Abemaciclib | FLT3(D835V) | 4.0 | 1000 | nM |
| Abemaciclib | FLT3(D835Y) | 96.0 | 100 | nM |
| Abemaciclib | FLT3(D835Y) | 31.0 | 1000 | nM |
| Abemaciclib | FLT3(ITD) | 100.0 | 100 | nM |
| Abemaciclib | FLT3(ITD) | 100.0 | 1000 | nM |
| Abemaciclib | FLT3(ITD,D835V) | 29.0 | 100 | nM |
| Abemaciclib | FLT3(ITD,D835V) | 5.1 | 1000 | nM |
| Abemaciclib | FLT3(ITD,F691L) | 71.0 | 100 | nM |
| Abemaciclib | FLT3(ITD,F691L) | 22.0 | 1000 | nM |
| Abemaciclib | FLT3(K663Q) | 100.0 | 100 | nM |
| Abemaciclib | FLT3(K663Q) | 74.0 | 1000 | nM |
| Abemaciclib | FLT3(N841I) | 79.0 | 100 | nM |
| Abemaciclib | FLT3(N841I) | 28.0 | 1000 | nM |
| Abemaciclib | FLT3(R834Q) | 100.0 | 100 | nM |
| Abemaciclib | FLT3(R834Q) | 100.0 | 1000 | nM |
| Abemaciclib | FLT3-autoinhibited | 76.0 | 100 | nM |
| Abemaciclib | FLT3-autoinhibited | 100.0 | 1000 | nM |